Sven Frøkjær
Professor, emeritus
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A calorimetric study of phosphocholine membranes mixed with desmopressin and its diacylated prodrug derivative (DPP)
Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 21 Feb 2002, In: International Journal of Pharmaceutics. 233, 1-2, p. 199-206 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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A helical structural nucleus is the primary elongating unit of insulin amyloid fibrils
Vestergaard, Bente, Jensen, M. G., Roessle, M., Kastrup, Jette Sandholm Jensen, van de Weert, Marco, Flink, J. M., Frøkjær, Sven, Gajhede, Michael & Svergun, D. I., 2007, In: PLoS - Biology. 5, 5, p. 1089-1097Research output: Contribution to journal › Journal article › Research › peer-review
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Assessment of side-chain modified dipeptides that interact with the oligopeptide transporter
Frøkjær, Sven, Steffansen, B. & Taub, M. E., 1998, Peptide and Protein Drug Delivery: Alfred Benzon Symposium 43. Munkgaard, p. 287-297 10 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Association of acylated cationic decapeptides with dipalmitoylphosphatidylserine-dipalmitoylphosphatidylcholine lipid membranes
Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 7 Nov 2001, In: Chemistry and Physics of Lipids. 113, 1-2, p. 83-95 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Association of an acylated model peptide with DPPC-DPPS lipid membranes
Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 77-81 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Beta-carboxylic acid esterfied D-Asp-Ala retains a high affinity for the oligopeptide transporter in Caco-2 cell monolayers
Taub, M. E., Larsen, B. D., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 146, p. 205-212 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Binding mode of Thioflavin T in insulin amyloid fibrils
Jensen, M. G., Norrman, M., Flink, J. M., van de Weert, Marco, Bukrinsky, J. T., Schluckebier, G. & Frøkjær, Sven, 2007, In: Journal of Structural Biology. 159, 3, p. 483-497Research output: Contribution to journal › Journal article › Research › peer-review
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Biologiske lægemidler - fra molekyle til medicin
Nielsen, Hanne Mørck, Foged, Camilla, Jørgensen, Lene & Frøkjær, Sven, 2013, In: Lægemiddelforskning. p. 12-14Research output: Contribution to journal › Journal article › Research
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Biotechnology-based pharmaceuticals
Jørgensen, Lene, Nielsen, Hanne Mørck & Frøkjær, Sven, 2009, Modern pharmaceutics: applications and advances. Florence, A. T. & Siepmann, J. (eds.). 5 ed. New York: Informa Healthcare, Vol. 2. p. 259-293 (Drugs and the Pharmaceutical Sciences, Vol. 188).Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
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Calcipotriol delivery into the skin with PEGylated liposomes
Knudsen, N. Ø., Rønholt, Stine, Salte, R. D., Jørgensen, Lene, Thormann, T., Basse, L. H., Hansen, J., Frøkjær, Sven & Foged, Camilla, 2012, In: European Journal of Pharmaceutics and Biopharmaceutics. 81, 3, p. 532-9 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Cellular uptake and membrane-destabilising properties of a-peptide/ß-peptoid chimeras: lessons for the design of new cell-penetrating peptides
Foged, Camilla, Franzyk, Henrik, Bahrami, S., Frøkjær, Sven, Jaroszewski, J. W., Nielsen, Hanne Mørck & Olsen, Christian Adam, 2008, In: BBA General Subjects. 1778, 11, p. 2487-2495Research output: Contribution to journal › Journal article › Research › peer-review
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Characterisation and physical stability of PEGylated glucagon
Stigsnæs, P., Frøkjær, Sven, Bjerregaard, S., van de Weert, Marco, Kingshott, P. & Møller, E. H., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 89-98Research output: Contribution to journal › Journal article › Research › peer-review
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Characterisation of salmon calcitonin in spray-dried powder for inhalation. Effect of chitosan
Yang, Mingshi, Velaga, S., Yamamoto, H., Takeuchi, H., Kawashima, Y., Hovgaard, L., van de Weert, Marco & Frøkjær, Sven, 2007, In: Internation Journal of Pharmaceutics. 331, 2, p. 176-181Research output: Contribution to journal › Journal article › Research › peer-review
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Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media
Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 2, p. 98-108 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Chemical and thermal stability of insulin: effects of zinc and ligand binding to the insulin zinc-hexamer
Huus, K., Havelund, S., Olsen, H. B., van de Weert, Marco & Frøkjær, Sven, Nov 2006, In: Pharmaceutical Research. 23, 11, p. 2611-20 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1
Søndergaard, H. B., Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2008, In: European Journal of Pharmaceutical Sciences. 33, 4-5, p. 332-342Research output: Contribution to journal › Journal article › Research › peer-review
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Complex coacervation of lysozyme and heparin: complex characterization and protein stability
van de Weert, Marco, Andersen, M. B. & Frøkjær, Sven, Dec 2004, In: Pharmaceutical Research. 21, 12, p. 2354-9 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Complex coacervation with heparin results in decreased lysozyme stability
van de Weert, Marco, Bendix Andersen, M. & Frøkjær, Sven, 3 Jan 2005, In: Journal of controlled release : official journal of the Controlled Release Society. 101, 1-3, p. 361-2 2 p.Research output: Contribution to journal › Conference abstract in journal › Research
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Computational prediction of solubilizers' effect on partitioning
Høst, J., Christensen, I. T., Jørgensen, Flemming Steen, Frøkjær, Sven & Hovgaard, L., 2007, In: Internation Journal of Pharmaceutics. 329, 1-2, p. 46-52Research output: Contribution to journal › Journal article › Research › peer-review
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Danish Physicians’ Views on the Appropriateness of the Involvement of Patients with Type 2 Diabetes in Regulatory Decision Making: A Qualitative Study
Sachs, M. L., Colding-Jørgensen, M., Helboe, P., Kälvemark Sporrong, Sofia, Frøkjær, Sven, Jelic, K. & Kaae, Susanne, 2019, In: Pharmaceutical Medicine. 33, 2, p. 99-107Research output: Contribution to journal › Journal article › Research › peer-review
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Data-enriched edible pharmaceuticals (DEEP) of medical cannabis by inkjet printing
Öblom, H., Cornett, Claus, Bøtker, Johan Peter, Frøkjær, Sven, Hansen, Harald S., Rades, Thomas, Rantanen, Jukka & Genina, Natalja, 2020, In: International Journal of Pharmaceutics. 589, p. 1-11 119866.Research output: Contribution to journal › Journal article › Research › peer-review
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Delivery aspects of small peptides and substrates for peptide transporters
Steffansen, B., Nielsen, C. U. & Frøkjær, Sven, 2005, In: European Journal of Pharmaceutics and Biopharmaceutics. 60, 4, p. 241-245 4 p.Research output: Contribution to journal › Review › Research › peer-review
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Den danske kodeks for integritet i forskning
Pedersen, H. M., Frøkjær, Sven, Bach, L. W., Vestergaard, E., Pedersen, C. V., Dirckinck-Holmfeld, L., Wegener, H. C., Jensen, L., Staunstrup, J. & Hansen, J. M., 2015Research output: Book/Report › Report › Communication
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Design of cyclic RKKH peptide-conjugated PEG liposomes targeting the integrin a2ß1 receptor
Knudsen, N. Ø., Schiffelers, R. M., Jørgensen, Lene, Hansen, J., Frøkjær, Sven & Foged, Camilla, 2012, In: International Journal of Pharmaceutics. 428, 1-2, p. 171-177Research output: Contribution to journal › Journal article › Research › peer-review
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Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line
Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven, Taub, M. E. & Steffansen, B., 2001, In: Journal of Controlled Release. 76, 1-2, p. 129-38 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Drug delivery by phospholipase A2 degradable liposomes
Davidsen, J., Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 67-69 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Drug delivery studies in Caco-2 monolayers V. Ethyl glucoside esters as a novel type of absorption enhancers
Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1 Mar 1996, In: S.T.P. Pharma Sciences. 6, 2, p. 157-161 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Drug delivery studies in Caco-2 monolayers. IV. Ethyl glycoside esters as a novel type of absorption enhancers.
Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1996, In: STP pharma sciences. p. 157-161Research output: Contribution to journal › Journal article › Research › peer-review
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Effects of sucrose on rFVIIa aggregation and methionine oxidation
Soenderkaer, S., Carpenter, J. F., van de Weert, Marco, Hansen, L. L., Flink, J. & Frøkjær, Sven, Apr 2004, In: European Journal of Pharmaceutical Sciences. 21, 5, p. 597-606 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Enzymatic degradation of polymer covered SOPC-liposomes in relation to drug delivery
Davidsen, Johan, Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 29 Jan 2001, In: Advances in Colloid and Interface Science. 89-90, p. 303-311 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2
Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 2004, In: American Journal of Physiology - Renal Physiology. 286, 2, p. 385-393Research output: Contribution to journal › Journal article › Research › peer-review
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Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line
Nielsen, C. U., Amstrup, J., Steffansen, B., Frøkjær, Sven & Larsen, Birger Brodin, 2001, In: American Journal of Physiology: Gastrointestinal and Liver Physiology. 281, 1, p. G191-9Research output: Contribution to journal › Journal article › Research › peer-review
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Erratum: Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: Affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism (Journal of Controlled Release (2003) 86 (279-292) PII: S0168365902004133)
Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 7 Mar 2003, In: Journal of Controlled Release. 88, 2Research output: Contribution to journal › Journal article › Research › peer-review
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Evaluation of statistical design/modeling for prediction of the effect of amino acids on agitation-induced aggregation of human growth hormone and human insulin
Soenderkaer, S., van de Weert, Marco, Lindgaard Hansen, L., Flink, J. & Frøkjær, Sven, 2005, In: Journal of Drug Delivery Science and Technology. 15, 6, p. 427-434 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Factors of importance for a successful delivery system for proteins
van de Weert, Marco, Jørgensen, Lene, Horn Moeller, E. & Frøkjær, Sven, Nov 2005, In: Expert Opinion on Drug Delivery. 2, 6, p. 1029-37 9 p.Research output: Contribution to journal › Review › Research › peer-review
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Formation mechanism of insulin fibrils and structural aspects of the insulin fibrillation process
Jensen, M. G., Frøkjær, Sven & Vestergaard, Bente, 2009, In: Current Protein and Peptide Science. 10, 5, p. 509-528Research output: Contribution to journal › Journal article › Research › peer-review
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Formulation, stability and characterization of protein and peptide drugs
Frøkjær, Sven, Hovgaard, L. & van de Weert, Marco, 2004, Biomaterials for Delivery and Targeting of Proteins and Nucleic Acids. Mahato, R. I. (ed.). Boca Raton: CRC Press, p. 378-401Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Communication
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Gennembrud i forståelsen af insulinfibrillering
Jensen, M. G., Vestergaard, Bente, Frøkjær, Sven, Gajhede, Michael, Flink, J. M., van de Weert, Marco, Kastrup, Jette Sandholm Jensen & Svergun, D. I., 2007, In: Lægemiddelforskning. p. 10-11Research output: Contribution to journal › Journal article › Communication
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Guidance for pediatric use in prescription information for novel medicinal products in the EU and the US
Christiansen, H., De Bruin, M. L., Frøkjær, Sven & Hallgreen, Christine Erikstrup, 2022, In: PLoS ONE. 17, 4, 19 p., e0266353.Research output: Contribution to journal › Journal article › Research › peer-review
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Human peptide transporters: Therapeutic applications
Nielsen, C. U., Larsen, Birger Brodin, Jørgensen, Flemming Steen, Frøkjær, Sven & Steffansen, B., 1 Sep 2002, In: Expert Opinion on Therapeutic Patents. 12, 9, p. 1329-1350 22 p.Research output: Contribution to journal › Journal article › Research › peer-review
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I-125 used for labelling of proteins in an absorption model changes the absorption rate of insulin aspart
Søhoel, A., Plum, A., Frøkjær, Sven & Thygesen, P., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 114-120Research output: Contribution to journal › Journal article › Research › peer-review
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In vitro and in vivo aspects of N-acyl-phosphatidylethanolamine-containing liposomes
Vermehren, Charlotte, Clausen-Beck, B., Frøkjær, Sven & Hansen, Harald S., 18 Mar 2003, In: International Journal of Pharmaceutics. 254, 1, p. 49-53 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
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In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1
Andersen, R., Nielsen, C. U., Begtrup, M., Jørgensen, Flemming Steen, Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2006, In: European Journal of Pharmaceutical Sciences. 28, 4, p. 325-35 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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In vitro release of insulin aspart incorporated into water-in-oil emulsions
Jørgensen, Lene, Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2004, In: Journal of Drug Delivery Science and Technology. 14, 6, p. 455-459Research output: Contribution to journal › Journal article › Research › peer-review
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In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model
Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 1 Jan 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 77-86 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Influence of PEGylation with linear and branched PEG chains on the adsorption of glucagon to hydrophobic surfaces
Pinholt, C., Bukrinsky, J. T., Hostrup, S., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 77, 1, p. 139-147Research output: Contribution to journal › Journal article › Research › peer-review
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Influence of acylation on the adsorption of GLP-2 to hydrophobic surfaces
Pinholt, C., Kapp, S. J., Bukrinsky, J. T., Hostrup, S., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2013, In: International Journal of Pharmaceutics. 440, 1, p. 63-71 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Influence of acylation on the adsorption of insulin to hydrophobic surfaces
Pinholt, C., Hostrup, S., Bukrinsky, J. T., Frøkjær, Sven & Jørgensen, Lene, 2011, In: Pharmaceutical Research. 28, p. 1031-1040Research output: Contribution to journal › Journal article › Research › peer-review
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Influence of glycosylation on the adsorption of Thermomyces lannuginosus lipase to hydrophobic and hydrophilic surfaces
Pinholt, C., Fanø, M., Wiberg, C., Hostrup, S., Bukrinsky, J. T., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2010, In: European Journal of Pharmaceutical Sciences. 40, 4, p. 273-281Research output: Contribution to journal › Journal article › Research › peer-review
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Influence of oligopeptide transporter binding affinity upon uptake and transport of D-Asp(Obzl)-Ala and Asp(OBzl)-Sar in filter-grown Caco-2 monolayers
Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 156, p. 219-228 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Interaction of dendritic cells with antigen-containing liposomes: effect of bilayer composition
Foged, Camilla, Arigita, C., Sundblad, A., Jiskoot, W., Storm, G. & Frøkjær, Sven, 2004, In: Vaccine. 22, 15-16, p. 1903-13 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Interfacial adsorption of insulin - conformational changes and reversibility of adsorption
Mollmann, S. H., Jørgensen, Lene, Bukrinsky, J. T., Elofsson, U., Norde, W. & Frøkjær, Sven, 2006, In: European Journal of Pharmaceutical Sciences. 27, 2-3, p. 194-204Research output: Contribution to journal › Journal article › Research › peer-review
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Intestinal solute carriers: an overview of trends and strategies for improving oral drug absorption
Steffansen, B., Nielsen, C. U., Larsen, Birger Brodin, Eriksson, A. H., Andersen, R. & Frøkjær, Sven, 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 3-16 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Ionic strength-dependent denaturation of Thermomyces lanuginosus lipase induced by SDS
Fanø, M., van de Weert, Marco, Møller, E. H., Kruse, N. A. & Frøkjær, Sven, 2011, In: Archives of Biochemistry and Biophysics. 506, 1, p. 92-98Research output: Contribution to journal › Journal article › Research › peer-review
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Issues in Development of Biodrug Delivery Systems
Jørgensen, Lene, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, Biodrug Delivery Systems: Fundamentals, Applications and Clinical Development. Morishita, M. & Park, K. (eds.). 1 ed. Informa Healthcare, p. 13-25Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Issues in development of biodrug delivery systems
Jørgensen, Lene, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, Biodrug delivery systems: fundamentals, applications and clinical development. Morishita, M. & Park, K. (eds.). New York: Informa Healthcare, p. 13-25Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
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Kinetics of insulin adsorption and gelation at the oil-water interface monitored using fluorescence correlation spectroscopy
Donsmark, J., Jørgensen, Lene, Mollmann, S. H., Frøkjær, Sven & Rischel, C., 2006, In: Pharmaceutical Research. 23, 1, p. 148-155Research output: Contribution to journal › Journal article › Research › peer-review
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Kinetics of insulin adsorption at the oil-water interface and diffusion properties of adsorbed layers monitored using fluorescence correlation spectroscopy
Donsmark, J., Jørgensen, Lene, Mollmann, S., Frøkjær, Sven & Rischel, C., 1 Jan 2006, In: Pharmaceutical Research. 23, 1, p. 148-155 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Ligand binding and thermostability of different allosteric states of the insulin zinc-hexamer
Huus, K., Havelund, S., Olsen, H. B., Sigurskjold, B. W., van de Weert, Marco & Frøkjær, Sven, 28 Mar 2006, In: Biochemistry. 45, 12, p. 4014-4024 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Liposomes for phospholipase A2 triggered siRNA release: preparation and in vitro test
Foged, Camilla, Nielsen, Hanne Mørck & Frøkjær, Sven, 2007, In: Internation Journal of Pharmaceutics. 331, 2, p. 160-166Research output: Contribution to journal › Journal article › Research › peer-review
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Medicon Valley - dansk-svensk succes
Jørgensen, S., Ahren, B., Jensen, I. S. & Frøkjær, Sven, 14 Mar 2013, In: Morgenavisen Jyllands-Posten. p. 28Research output: Contribution to journal › Contribution to newspaper - Feature article › Communication
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Metode til screening af modificerede proteinlægemidler under opbevaring
Petersen, C., Jørgensen, Lene, Hostrup, S., Bukrinsky, J. T. & Frøkjær, Sven, 2008, In: Lægemiddelforskning. p. 16-18Research output: Contribution to journal › Journal article › Communication
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Micropipette manipulation a technique to evaluate the stability of water-in-oil emulsions containing proteins
Jørgensen, Lene, Kim, D. H., Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2004, In: Journal of Pharmaceutical Sciences. 93, 12, p. 2994-3003Research output: Contribution to journal › Journal article › Research › peer-review
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Model prodrugs for the intestinal oligopeptide transporter: model drug release in aqueous solution and in various biological media
Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2001, In: Journal of Controlled Release. 73, 1, p. 21-30 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Novel formulation approaches for peptide and protein injectables
Yang, Mingshi & Frøkjær, Sven, 2009, Delivery technologies for biopharmaceuticals: Peptides, proteins, nucleic acids and vaccines. Jørgensen, L. & Mørck Nielsen, H. (eds.). Wiley, p. 11-28Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
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Oligopeptide transporter mediated uptake and transport of D-Asp(OBzl)-Ala, D-Glu(OBzl)-Ala and D-Ser(Bzl)-Ala in filter grown Caco-2 monolayers
Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1998, In: International Journal of Pharmaceutics. 174, p. 223-232 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Particle size and surface charge affect particle uptake by human dendritic cells in an in vitro model
Foged, Camilla, Larsen, Birger Brodin, Frøkjær, Sven & Sundblad, A., 2005, In: Internation Journal of Pharmaceutics. 298, 2, p. 315-22 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Penetration of gel and liquid state liposomes into barrier-impaired skin
Knudsen, N. Ø., Frøkjær, Sven, Hansen, J., Jørgensen, Lene & Foged, Camilla, 2010, In: Journal of Pharmacy and Pharmacology. p. 793Research output: Contribution to journal › Conference article › Research › peer-review
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Peptide and protein drug delivery : proceedings of a symposium held at the Royal Danish Academy of Sciences and Letters, August 17-21, 1997: Alfred Benzon Symposium, 43
Frøkjær, Sven, Christrup, Lona Louring, Krogsgaard-Larsen, Povl & Alfred Benzon, F., 1998, Copenhagen: Munksgaard .Research output: Book/Report › Book › Research
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Phase behavior and lipid-membrane structure of phospholipid- glycosphingolipid liposomes and the thermal unfolding of insulin
Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 1 Jan 1999, In: Journal of Liposome Research. 9, 2, p. 261-274 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Phase behavior and nanoscale structure of phospholipid membranes incorporated with acylated C14-peptides
Pedersen, T. B., Kaasgaard, T., Jensen, M., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., Oct 2005, In: Biophysical Journal. 89, 4, p. 2494-2503 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Phospholipase A2 sensitive liposomes for delivery of small interfering RNA (siRNA)
Foged, Camilla, Nielsen, Hanne Mørck & Frøkjær, Sven, 2007, In: Journal of Liposome Research. 17, 3-4Research output: Contribution to journal › Journal article › Research › peer-review
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Preparation and characterization of poly (DL-lactide-co-glycolide) nanoparticles for siRNA delivery
Cun, D., Foged, Camilla, Yang, Mingshi, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, In: Internation Journal of Pharmaceutics. 390, 1, p. 70-75Research output: Contribution to journal › Journal article › Research › peer-review
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Preparing and evaluating delivery systems for proteins
Jorgensen, L., Moeller, E. H., van de Weert, Marco, Nielsen, H. M. & Frøkjær, Sven, 2006, In: European Journal of Pharmaceutical Sciences. 29, 3-4, p. 174-82 9 p.Research output: Contribution to journal › Review › Research › peer-review
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Probing structural changes of proteins incorporated into water-in-oil emulsions
Jørgensen, Lene, van de Weert, Marco, Vermehren, C., Bjerregaard, S. & Frøkjær, Sven, Jul 2004, In: Journal of Pharmaceutical Sciences. 93, 7, p. 1847-59 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Prodrugs
Steffansen, B., Thomsen, A. E. & Frøkjær, Sven, 2003, Estimation of solubility, permeability, absorption and bioavaibility. van de Waterbeemd, H., Lennernäs, H. & Artursson, P. (eds.). Weinheim: Wiley-VCH, p. 532-546Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
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Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism
Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 2003, In: Journal of Controlled Release. 86, 2-3, p. 279-92 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Risk Perceptions in Diabetic Patients Who Have Experienced Adverse Events: Implications for Patient Involvement in Regulatory Decisions
Sachs, M. L., Kälvemark Sporrong, Sofia, Colding-Jørgensen, M., Frøkjær, Sven, Helboe, P., Jelic, K. & Kaae, Susanne, 2017, In: Pharmaceutical Medicine. 31, 4, p. 245-255 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Secondary structure alteration in insulin and growth hormone water-in-oil emulsions
Jørgensen, Lene, Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2003, In: Internation Journal of Pharmaceutics. 254, 1, p. 7-10Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Spray drying of siRNA-containing PLGA nanoparticles intended for inhalation
Jensen, D. M. K., Cun, D., Maltesen, M. J., Frøkjær, Sven, Nielsen, Hanne Mørck & Foged, Camilla, 2010, In: Journal of Controlled Release. 142, p. 138-145Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Stability and vitro metabolism of dipeptide model prodrugs with affinity for the oligopeptide transporter
Lepist, E., Steffansen, B., Kusk, T., Larsen, D. H., Andersen, D., Frøkjær, Sven, Taub, M. E., Veski, P. & Lennernas, H., 2000, In: European Journal of Pharmaceutical Sciences. 11, p. 43-50 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Stability metabolism and transport of D-Asp(OBzl)Ala -a model prodrug with affinity for the oligopeptide transporter
Steffansen, B., Lepist, E., Frøkjær, Sven, Taub, M. E. & Lennernas, H., 1999, In: European Journal of Pharmaceutical Sciences. 8, p. 67-73Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Study on the binding of Thioflavin T to ß-sheet-rich and non-ß-sheet cavities
Jensen, M. G., Olsen, L., van de Weert, Marco, Flink, J. M., Frøkjær, Sven & Jørgensen, Flemming Steen, 2007, In: Journal of Structural Biology. 158, 3, p. 358-369Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Targeting of liposome-associated calcipotriol to the skin: effect of liposomal membrane fluidity and skin barrier integrity
Knudsen, N. Ø., Jørgensen, Lene, Hansen, J., Vermehren, C., Frøkjær, Sven & Foged, Camilla, 2011, In: International Journal of Pharmaceutics. 416, p. 478-485Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The effect of beta-turn structure on the permeation of peptides across monolayers of bovine brain microvessel endothelial cells
Sørensen, M., Steenberg, B., Knipp, G., Wang, W., Steffansen, B., Frøkjær, Sven & Borchardt, R. T., 1997, In: Pharmaceutical Research. 14, p. 1341-1348Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The novel oxygenated chalcone, 2,4-dimethoxy-4'-butoxychalcone, exhibits potent activity against human malaria parasite Plasmodium falciparum in vitro and rodent parasites Plasmodium berghei and Plasmodium yoelii in vivo
Chen, M., Christensen, Søren Brøgger, Zhai, L., Rasmussen, M. H., Theander, Thor Grundtvig, Frøkjær, Sven, Steffansen, B., Davidsen, J. & Kharazmi, A., 1997, In: Journal of Infectious Diseases. 176, 5, p. 1327-33 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Thermal dissociation and unfolding of insulin
Huus, K., Havelund, S., Olsen, H. B., van de Weert, Marco & Frøkjær, Sven, 23 Aug 2005, In: Biochemistry. 44, 33, p. 11171-7 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line
Nielsen, C. U., Supuran, C. T., Scozzafava, A., Frøkjær, Sven, Steffansen, B. & Larsen, Birger Brodin, 2002, In: Pharmaceutical Research. 19, 9, p. 1337-44 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1
Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B. & Frøkjær, Sven, 2002, In: Basic & Clinical Pharmacology & Toxicology. 90, 6, p. 285-96 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Risk Perceptions in Diabetic Patients Who Have Experienced Adverse Events: Implications for Patient Involvement in Regulatory Decisions
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Guidance for pediatric use in prescription information for novel medicinal products in the EU and the US
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