Lasse Saaby
Affiliated Associate Professor, Guest Researcher
- 2008
- Published
MAO-A inhibitory activity of quercetin from Calluna vulgaris Hull
Saaby, Lasse, Jäger, A. K. & Rasmussen, H. B., 2008.Research output: Contribution to conference › Poster › Research
- 2009
- Published
MAO-A inhibitory activity of quercetin from Calluna vulgaris (L.) Hull
Saaby, Lasse, Rasmussen, H. B. & Jäger, A. K., 2009, In: Journal of Ethnopharmacology. 121, 1, p. 178-181Research output: Contribution to journal › Journal article › Research › peer-review
- 2010
- Published
Short communication: Influence of pasteurization on the active compounds in medicinal plants to be used in dairy products
Jäger, A. K., Saaby, Lasse, Kudsk, D. S., Witt, K. C. & Mølgaard, Per, 2010, In: Journal of Dairy Science. 93, 6, p. 2351-2353Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Characterization of anti-inflammatory triterpene acids from rose hip powder (Rosa canina L.)
Saaby, Lasse, Jäger, A., Moesby, L., Hansen, E. W. & Christensen, Søren Brøgger, Aug 2010, In: Planta Medica. 76, 12, p. 1171Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
- 2011
- Published
Evaluation of immunomodulating and anti-inflammatory effects of a herbal remedy based on rose hip powder (Rosa canina L.)
Saaby, Lasse, 2011, København: Det Farmaceutiske Fakultet. 130 p.Research output: Book/Report › Ph.D. thesis › Research
- Published
Isolation of immunomodulatory triterpene acids from a standardized rose hip powder (Rosa canina L.)
Saaby, Lasse, Jäger, A. K., Moesby, L., Hansen, E. W. & Christensen, Søren Brøgger, Feb 2011, In: Phytotherapy Research. 25, 2, p. 195-201Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Flavonoids and the CNS
Jäger, A. K. & Saaby, Lasse, 10 Feb 2011, In: Molecules. 16, 2, p. 1471-1485Research output: Contribution to journal › Review › Research › peer-review
- Published
Ubiquitous plant compounds disturb cell-based assays
Saaby, Lasse & Jäger, A. K., 1 Sep 2011, In: Journal of Ethnopharmacology. 137, 1, p. 942-943Research output: Contribution to journal › Comment/debate › Research › peer-review
- 2012
- Published
Triterpene Acids from Rose Hip Powder Inhibit Self-antigen- and LPS-induced Cytokine Production and CD4(+) T-cell Proliferation in Human Mononuclear Cell Cultures
Saaby, Lasse & Nielsen, Claus Henrik, Aug 2012, In: Phytotherapy Research. 26, 8, p. 1142-1147 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2013
- Published
Current status of rational design of prodrugs targeting the intestinal di/tri-peptide transporter hPEPT1 (SLC15A1)
Saaby, Lasse, Nielsen, C. U., Steffansen, B., Larsen, Birger Brodin & Larsen, S. B. L., 2013, In: Journal of Drug Delivery Science and Technology. 23, 4, p. 307–314Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Considerations regarding use of solvents in in vitro cell based assays
Timm, M., Saaby, Lasse, Moesby, L. & Hansen, E. W., Oct 2013, In: Cytotechnology. 65, 5, p. 887-894 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Bioavailability of cinnarizine in dogs: effect of SNEDDS loading level and correlation with cinnarizine solubilization during in vitro lipolysis
Larsen, A. T., Åkesson, P., Juréus, A., Saaby, Lasse, Abu-Rmaileh, R., Abrahamsson, B., Østergaard, Jesper & Mullertz, Anette , Dec 2013, In: Pharmaceutical Research. 30, 12, p. 3101-13 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2014
- Published
THE POSSIBLE EFFECT OF TELMISARTAN ON THE BLOOD-BRAIN BARRIER TRANSPORT OF VERAPAMIL.
Saaby, Lasse, Tfelt-Hansen, P. & Larsen, Birger Brodin, 18 Sep 2014. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- 2015
- Published
Characterization of particulate drug delivery systems for oral delivery of Peptide and protein drugs
Christophersen, P. C., Fano, M., Saaby, Lasse, Yang, Mingshi, Nielsen, Hanne Mørck & Mu, Huiling, 2015, In: Current Pharmaceutical Design. 21, 19, p. 2611-28 18 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The putative P-gp inhibitor telmisartan does not affect the transcellular permeability and cellular uptake of the calcium channel antagonist verapamil in the P-glycoprotein expressing cell line MDCK II MDR1
Saaby, Lasse, Tfelt-Hansen, P. & Larsen, Birger Brodin, 11 Jun 2015, In: Pharmacology Research & Perspectives. 3, 4, p. 1-9 9 p., e00151.Research output: Contribution to journal › Journal article › Research › peer-review
- 2016
- Published
Survival of Lactobacillus acidophilus NCFM® and Bifidobacterium lactis HN019 encapsulated in chocolate during in vitro simulated passage of the upper gastrointestinal tract
Klindt-Toldam, S., Larsen, S. K., Saaby, Lasse, Olsen, L. R., Svenstrup, G., Mullertz, Anette , Knoechel, Susanne, Heimdal, H., Nielsen, Dennis Sandris & Zielińska, D., 2016, In: Lebensmittel - Wissenschaft und Technologie. 74, p. 404-410 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
IPEC-J2 MDR1, a Novel High-Resistance Cell Line with Functional Expression of Human P-glycoprotein (ABCB1) for Drug Screening Studies
Saaby, Lasse, Helms, H. C. C. & Larsen, Birger Brodin, 1 Feb 2016, In: Molecular Pharmaceutics. 13, 2, p. 640-52 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Apomorphine and its esters: Differences in Caco-2 cell permeability and chylomicron affinity
Borkar, N., Chen, Z., Saaby, Lasse, Mullertz, Anette , Håkansson, A. E., Schönbeck, C., Yang, Mingshi, Holm, R. & Mu, Huiling, 6 Jun 2016, In: International Journal of Pharmaceutics. 509, 1-2, p. 499–506 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Development of a μDissolution-Permeation model with in situ drug concentration monitoring
Berthelsen, R., Byrialsen, J. P., Holm, R., Jacobsen, Jette, Abrahamsson, B., Saaby, Lasse, Madelung, P. & Mullertz, Anette , 1 Oct 2016, In: Journal of Drug Delivery Science and Technology. 35, p. 223-233 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2017
- Published
iP-gp , a novel cell line with tight barrier function and expression of human P-glycoprotein (ABCB1) for drug screening
Larsen, Birger Brodin, Ozgür, Burak & Saaby, Lasse, 23 May 2017.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
A Critical View on In Vitro Analysis of P-glycoprotein (P-gp) Transport Kinetics
Saaby, Lasse & Larsen, Birger Brodin, Sep 2017, In: Journal of Pharmaceutical Sciences. 106, 9, p. 2257-2264 8 p.Research output: Contribution to journal › Review › Research › peer-review
- 2018
- Published
Characterization of the IPEC-J2 MDR1 (iP-gp) cell line as a tool for identification of P-gp substrates
Ozgür, Burak, Saaby, Lasse, Langthaler, K. & Larsen, Birger Brodin, 2018, In: European Journal of Pharmaceutical Sciences. 112, p. 112-121 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Data demonstrating the challenges of determining the kinetic parameters of P-gp mediated transport of low-water soluble substrates
Ozgür, Burak, Saaby, Lasse, Langthaler, K. & Larsen, Birger Brodin, 2018, In: Data in Brief. 16, p. 655-659 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Hydrolysed pea proteins mitigate in vitro wheat starch digiestibility
López-Barón , N., Sagnelli, D., Blennow, Andreas, Holse, M., Gao, J., Saaby, Lasse, Mullertz, Anette , Jespersen, Birthe P Møller & Vasanthan, T., Jun 2018, In: Food Hydrocolloids. 79, p. 117-126 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The iP-gp cell model is an improved tool for predicting the in vivo relevance of P-gp mediated efflux at the blood-brain barrier
Ozgür, Burak, Saaby, Lasse, Eneberg, E., Langthaler, K., Jacobsen, A., Janfelt, Christian, Badolo, L., Montanari, D. & Larsen, Birger Brodin, 22 Jun 2018.Research output: Contribution to conference › Poster › Research › peer-review
ID: 4863000
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Data demonstrating the challenges of determining the kinetic parameters of P-gp mediated transport of low-water soluble substrates
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
173
downloads
The Pyrazolo[3,4-d]pyrimidine Derivative, SCO-201, Reverses Multidrug Resistance Mediated by ABCG2/BCRP
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
67
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A novel derivative of thioridazine shows low toxicity and efficient activity against gram‐positive pathogens
Research output: Contribution to journal › Journal article › Research › peer-review
Published