Physiological Pharmaceutics

  1. 2019
  2. Published

    Ex vivo intestinal perfusion model for investigating mucoadhesion of microcontainers

    Dalskov Mosgaard, M., Strindberg, S., Abid, Z., Singh Petersen, R., Højlund Eklund Thamdrup, L., Joukainen Andersen, A., Sylvest Keller, S., Mullertz, Anette , Hagner Nielsen, L. & Boisen, A., 2019, In: International Journal of Pharmaceutics. 570, 118658.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Quantification of Inkjet-Printed Pharmaceuticals on Porous Substrates Using Raman Spectroscopy and Near-Infrared Spectroscopy

    Edinger, M., Iftimi, L., Markl, D., Al-Sharabi, M., Bar-Shalom, Daniel, Rantanen, Jukka & Genina, Natalja, Jul 2019, In: AAPS PharmSciTech. 20, 5, 10 p., 207.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Mimicking regional and fasted/fed state conditions in the intestine with the mucus-PVPA in vitro model: The impact of pH and simulated intestinal fluids on drug permeability

    Falavigna, M., Klitgaard, Mette, Steene, E. & Flaten, G. E., 30 Apr 2019, In: European Journal of Pharmaceutical Sciences. 132, p. 44-54 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Visualization of the penetration modifying mechanism of laurocapram by Mass Spectrometry Imaging in buccal drug delivery

    Handler, A. M., Marxen, E., Jacobsen, Jette & Janfelt, Christian, 15 Jan 2019, In: European Journal of Pharmaceutical Sciences. 127, p. 276-281 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Edible solid foams as porous substrates for inkjet-printable pharmaceuticals

    Iftimi, L., Edinger, M., Bar-Shalom, Daniel, Rantanen, Jukka & Genina, Natalja, Mar 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 136, p. 38-47

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Fast and quantitative 2D and 3D orientation mapping using Raman microscopy

    Ilchenko, O., Pilgun, Y., Kutsyk, A., Slipets, R., Bachmann, F., Todeschini, M., Okeyo, P. O., Friis Poulsen, H. & Boisen, A., 5 Dec 2019, In: Nature Communications. 10, 9 p., 5555.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Exploring the utility of the Chasing-rinciple: influence of drug-free SNEDDS composition on solubilization of carvedilol, cinnarizine and R3040 in aqueous suspension

    Jorgensen, S. D. S., Rades, Thomas, Mu, Huiling, Graeser, K. & Mullertz, Anette , Jan 2019, In: Acta Pharmaceutica Sinica B. 9, 1, p. 194-201

    Research output: Contribution to journalLetterResearchpeer-review

  9. Published

    Determining Thermal Conductivity of Small Molecule Amorphous Drugs with Modulated Differential Scanning Calorimetry and Vacuum Molding Sample Preparation

    Karl, M., Rantanen, Jukka & Rades, Thomas, 6 Dec 2019, In: Pharmaceutics. 11, 12, 7 p., 670.

    Research output: Contribution to journalJournal articleCommunication

  10. Published

    SEDDS for intestinal absorption of insulin: Application of Caco-2 and Caco-2/HT29 co-culture monolayers and intra-jejunal instillation in rats

    Liu, J., Werner, U., Funke, M., Besenius, M., Saaby, Lasse, Fano, M., Mu, Huiling & Mullertz, Anette , 5 Apr 2019, In: International Journal of Pharmaceutics. 560, p. 377-384

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Polymeric Lids for Microcontainers for Oral Protein Delivery

    Mazzoni, C., Jacobsen, R. D., Mortensen, J., Jørgensen, J. R., Vaut, L., Jacobsen, Jette, Gundlach, C., Mullertz, Anette , Nielsen, L. H. & Boisen, A., 2019, In: Macromolecular Bioscience. 19, 5, 1900004.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Fenofibrate oral absorption from SNEDDS and super-SNEDDS is not significantly affected by lipase inhibition in rats

    Michaelsen, M. H., Siqueira Jørgensen, S. D., Abdi, I. M., Wasan, K. M., Rades, Thomas & Mullertz, Anette , 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 142, p. 258-264 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Imaging of dehydration in particulate matter using Raman line-focus microscopy

    Okeyo, P. O., Ilchenko, O., Slipets, R., Larsen, P. E., Boisen, A., Rades, Thomas & Rantanen, Jukka, 17 May 2019, In: Scientific Reports. 9, 11 p., 7525.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Digestive Enzyme Corona Formed in the Gastrointestinal Tract and Its Impact on Epithelial Cell Uptake of Nanoparticles

    Peng, Q., Liu, J., Zhang, T., Zhang, T., Zhang, C. & Mu, Huiling, 8 Apr 2019, In: Biomacromolecules. 20, 4, p. 1789-1797 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Microcontainers for oral insulin delivery - in vitro studies of permeation enhancement

    Rune Jørgensen, J., Leth Jepsen, M., Hagner Nielsen, L., Dufva, M., Nielsen, Hanne Mørck, Rades, Thomas, Boisen, A. & Mullertz, Anette , 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 143, p. 98-105

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Acids ‘generally recognized as safe’ affect morphology and biocompatibility of electrospun chitosan/polyethylene oxide nanofibers

    Stie, Mai Bay, Jones, M., Sørensen, H. O., Jacobsen, Jette, Chronakis, I. S. & Nielsen, Hanne Mørck, 1 Jul 2019, In: Carbohydrate Polymers. 215, p. 253-262

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    A Bayesian Generative Model with Gaussian Process Priors for Thermomechanical Analysis of Micro-Resonators

    Vording, M. F., Okeyo, P. O., Guillamon, J. J. R., Larsen, P. E., Schmidt, M. N. & Alstrom, T. S., 2019, 2019 IEEE 29th International Workshop on Machine Learning for Signal Processing, MLSP 2019. IEEE, 8918876. (IEEE International Workshop on Machine Learning for Signal Processing, MLSP, Vol. 2019-October).

    Research output: Chapter in Book/Report/Conference proceedingArticle in proceedingsResearchpeer-review

  18. Published

    In vivo models and decision trees for formulation development in early drug development: A review of current practices and recommendations for biopharmaceutical development

    Zane, P., Gieschen, H., Kersten, E., Mathias, N., Ollier, C., Johansson, P., Van den Bergh, A., Van Hemelryck, S., Reichel, A., Rotgeri, A., Schäfer, K., Mullertz, Anette & Langguth, P., 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 142, p. 222-231 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. 2020
  20. Published

    Six years of progress in the oral biopharmaceutics area – A summary from the IMI OrBiTo project

    Abrahamsson, B., Mcallister, M., Augustijns, P., Zane, P., Butler, J., Holm, R., Langguth, P., Lindahl, A., Mullertz, Anette , Pepin, X., Rostami-hodjegan, A., Sjögren, E., Berntsson, M. & Lennernäs, H., 1 Jul 2020, In: European Journal of Pharmaceutics and Biopharmaceutics. 152, p. 236-247 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Direct Measurement of Lateral Molecular Diffusivity on the Surface of Supersaturated Amorphous Solid Dispersions by Atomic Force Microscopy

    Bannow, J., Karl, M., Larsen, P. E., Hwu, E. T. & Rades, Thomas, 2020, In: Molecular Pharmaceutics. 17, 5, p. 1715-1722 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Improving the drug load and in vitro performance of supersaturated self-nanoemulsifying drug delivery systems (super-SNEDDS) using polymeric precipitation inhibitors

    Bannow, J., Yorulmaz, Y., Löbmann, Korbinian, Mullertz, Anette & Rades, Thomas, 2020, In: International Journal of Pharmaceutics. 575, 1188960.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    An Ingestible Self-Polymerizing System for Targeted Sampling of Gut Microbiota and Biomarkers

    Chen, L., Gruzinskyte, L., Jorgensen, S. L., Boisen, A. & Srivastava, S. K., 2020, In: ACS Nano. 14, 9, p. 12072-12081 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Milk osteopontin retains integrin-binding activity after in vitro gastrointestinal transit

    Christensen, B., Karlsen, N. J., Jorgensen, S. D. S., Jacobsen, L. N., Ostenfeld, M. S., Petersen, S. V., Mullertz, Anette & Sorensen, E. S., Jan 2020, In: Journal of Dairy Science. 103, 1, p. 42-51

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Fabrication of Mucoadhesive Buccal Films for Local Administration of Ketoprofen and Lidocaine Hydrochloride by Combining Fused Deposition Modeling and Inkjet Printing

    Eleftheriadis, G. K., Monou, P. K., Bouropoulos, N., Bøtker, Johan Peter, Rantanen, Jukka, Jacobsen, Jette, Vizirianakis, I. S. & Fatouros, D. G., 2020, In: Journal of Pharmaceutical Sciences. 109, 9, p. 2757-2766

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Evaluating side-by-side diffusion models for studying drug supersaturation in an absorptive environment: a case example of fenofibrate and felodipine

    Eliasen, Jannik Nicklas, Berthelsen, R., Slot, A. L. & Mullertz, Anette , 2020, In: Journal of Pharmacy and Pharmacology. 72, 3, p. 371-384

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Microenvironmental pH modifying films for buccal delivery of saquinavir: Effects of organic acids on pH and drug release in vitro

    He, S., Østergaard, Jesper, Ashna, M., Nielsen, C. U., Jacobsen, Jette & Mu, Huiling, 2020, In: International Journal of Pharmaceutics. 585, 10 p., 119567.

    Research output: Contribution to journalJournal articleResearchpeer-review