Pharmaceutical Physical and Analytical Chemistry

  1. 2019
  2. Published

    Distribution of platinum between nuclear and cytosolic fractions: can subcellular fractionation be performed quantitatively?

    Dam, C. S., Lambert, Ian Henry, Gammelgaard, Bente & Stürup, Stefan, 2019, In: Journal of Pharmaceutical and Biomedical Analysis. 165, p. 82-89 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Ex vivo toxicological evaluation of experimental anticancer gold(I) complexes with lansoprazole-type ligands

    Estrada-Ortiz, N., Lopez-Gonzales, E., Woods, B., Stürup, Stefan, de Graaf, I. A. M., Groothuis, G. M. M. & Casini, A., 1 Nov 2019, In: Toxicology Research. 8, 6, p. 885-895

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Pyrolysis preparation of poly-gamma-glutamic acid derived amorphous carbon nitride for supporting Ag and gamma-Fe2O3 nanocomposites with catalytic and antibacterial activity

    Feng, J., Shi, Q., Li, Y., Huang, Jianfei, Li, R., Shu, X., Li, W. & Xie, X., Aug 2019, In: Materials Science and Engineering: A - Structural Materials: Properties, Microstructure and Processing. 101, p. 138-147

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    From Structure to Function: pH-Switchable Antimicrobial Nano-Self-Assemblies

    Gontsarik, M., Yaghmur, Anan, Ren, Q., Maniura-Weber, K. & Salentinig, S., 27 Dec 2019, In: A C S Applied Materials and Interfaces. 11, 3, p. 2821–2829

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Development of a UPLC-IDA-ICP-MS/MS method for peptide quantitation in plasma by Se-labelling and comparison to S-detection of the native peptide

    Grønbæk-Thorsen, F., Stürup, Stefan, Gammelgaard, Bente & Møller, L. H., 2019, In: Journal of Analytical Atomic Spectrometry. 34, p. 375-383 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Exploring the utility of the Chasing-rinciple: influence of drug-free SNEDDS composition on solubilization of carvedilol, cinnarizine and R3040 in aqueous suspension

    Jorgensen, S. D. S., Rades, Thomas, Mu, Huiling, Graeser, K. & Mullertz, Anette , Jan 2019, In: Acta Pharmaceutica Sinica B. 9, 1, p. 194-201

    Research output: Contribution to journalLetterResearchpeer-review

  8. Published

    SEDDS for intestinal absorption of insulin: Application of Caco-2 and Caco-2/HT29 co-culture monolayers and intra-jejunal instillation in rats

    Liu, J., Werner, U., Funke, M., Besenius, M., Saaby, Lasse, Fano, M., Mu, Huiling & Mullertz, Anette , 5 Apr 2019, In: International Journal of Pharmaceutics. 560, p. 377-384

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Two-phase bipolar electrografting

    Madsen, M. R., Koefoed, L., Jensen, H., Daasbjerg, K. & Pedersen, S. U., 2019, In: Electrochimica Acta. 317, p. 61-69 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Transport characteristics in a novel in vitro release model for testing the performance of intra-articular injectables

    Mertz, Nina, Østergaard, Jesper, Yaghmur, Anan & Larsen, Susan Weng, 20 Jul 2019, In: International Journal of Pharmaceutics. 566, p. 445-453

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    The Interplay Between Blood Proteins, Complement, and Macrophages on Nanomedicine Performance and Responses

    Moghimi, S. M., Simberg, D., Skotland, T., Yaghmur, Anan & Hunter, A. C., 1 Sep 2019, In: Journal of Pharmacology and Experimental Therapeutics. 370, 3, p. 581-592

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Flow-Induced Dispersion Analysis (FIDA) for Protein Quantification and Characterization

    Pedersen, M. E., Østergaard, Jesper & Jensen, H., 2019, Clinical Applications of Capillary Electrophoresis. Springer, Vol. 1972. p. 109-123 15 p. (Methods in molecular biology (Clifton, N.J.)).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  13. Published

    Protein Characterization in 3D: Size, Folding and Functional Assessment in a Unified Approach

    Pedersen, M. E., Gad, S. I., Østergaard, Jesper & Jensen, H., 27 Mar 2019, In: Analytical Chemistry. 91, 8, p. 4975-4979

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Introduction to Pharmaceutical Analytical Chemistry

    Pedersen-Bjergaard, Stig, Gammelgaard, Bente & Grønhaug Halvorsen, T., 2019, 2 ed. Wiley. 544 p.

    Research output: Book/ReportBookEducationpeer-review

  15. Published

    Digestive Enzyme Corona Formed in the Gastrointestinal Tract and Its Impact on Epithelial Cell Uptake of Nanoparticles

    Peng, Q., Liu, J., Zhang, T., Zhang, T., Zhang, C. & Mu, Huiling, 8 Apr 2019, In: Biomacromolecules. 20, 4, p. 1789-1797 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Citrem-phosphatidylcholine nano-self-assemblies: solubilization of bupivacaine and its role in triggering a colloidal transition from vesicles to cubosomes and hexosomes

    Prajapati, R., Larsen, Susan Weng & Yaghmur, Anan, 21 Jul 2019, In: Physical Chemistry Chemical Physics. 21, 27, p. 15142-15150

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    pH-Responsive Nano-Self-Assemblies of the Anticancer Drug 2-Hydroxyoleic Acid

    Prajapati, R., Gontsarik, M., Yaghmur, Anan & Salentinig, S., 18 Jun 2019, In: Langmuir. 35, 24, p. 7954-7961

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Monitoring of antimicrobial drug chloramphenicol release from electrospun nano-and microfiber mats using UV imaging and bacterial bioreporters

    Preem, L., Bock, Frederik, Hinnu, M., Putrinš, M., Sagor, K., Tenson, T., Meos, A., Østergaard, Jesper & Kogermann, K., 2019, In: Pharmaceutics. 11, 9, 19 p., 487.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Electromembrane Extraction of Unconjugated Fluorescein Isothiocyanate from Solutions of Labeled Proteins Prior to Flow Induced Dispersion Analysis

    Restan, M. S., Pedersen, M. E., Jensen, H. & Pedersen-Bjergaard, Stig, 21 May 2019, In: Analytical Chemistry. 91, 10, p. 6702-6708

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Simulated synovial fluids for in vitro drug and prodrug release testing of depot injectables intended for joint injection

    Thing, M., Mertz, Nina, Ågårdh, L., Larsen, Susan Weng, Østergaard, Jesper & Larsen, C., 2019, In: Journal of Drug Delivery Science and Technology. 49, p. 169-176 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Electromembrane extraction with solvent modification of the acceptor solution: improved mass transfer of drugs of abuse from human plasma

    Vårdal, L., Øiestad, E. L., Gjelstad, A., Jensen, H. & Pedersen-Bjergaard, Stig, 2019, In: Bioanalysis. 11, p. 755-771

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    In vivo evaluation of solid lipid microparticles and hybrid polymer-lipid microparticles for sustained delivery of leuprolide

    Wu, C., Luo, X., Baldursdottir, S. G., Yang, Mingshi, Sun, X. & Mu, Huiling, 9 Jul 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 142, p. 315-321

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    A hydrodynamic flow focusing microfluidic device for the continuous production of hexosomes based on docosahexaenoic acid monoglyceride

    Yaghmur, Anan, Ghazal, A., Ghazal, R., Dimaki, M. & Svendsen, W. E., 28 Jun 2019, In: Physical chemistry chemical physics : PCCP. 21, 24, p. 13005-13013 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Internal Lamellar and Inverse Hexagonal Liquid Crystalline Phases During the Digestion of Krill and Astaxanthin Oil-in-Water Emulsions

    Yaghmur, Anan, Lotfi, S., Ariabod, S. A., Bor, G., Gontsarik, M. & Salentinig, S., 2019, In: Frontiers in Bioengineering and Biotechnology. 7, 12 p., 00384.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Nanoencapsulation of Food Ingredients by Cubosomes and Hexosomes

    Yaghmur, Anan, 2019, Lipid-Based Nanostructures for Food Encapsulation Purposes. Elsevier Ltd. Academic Press, Vol. 2. 483 p. (Elsevier Book Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  26. 2018
  27. Published

    Cisplatin Encapsulation Generates Morphologically Different Multicompartments in the Internal Nanostructures of Nonlamellar Liquid-Crystalline Self-Assemblies

    Azmi, I. D. M., Østergaard, Jesper, Stürup, Stefan, Gammelgaard, Bente, Urtti, A., Moghimi, S. M. & Yaghmur, Anan, 5 Jun 2018, In: Langmuir : the ACS journal of surfaces and colloids. 34, 22, p. 6570-6581 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Evaluation of drug permeation under fed state conditions using mucus-covered Caco-2 cell epithelium

    Birch, D., Diedrichsen, Ragna Guldsmed, Christophersen, P. C., Mu, Huiling & Nielsen, Hanne Mørck, Jun 2018, In: European Journal of Pharmaceutical Sciences. 118, p. 144-153

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    A fast and novel internal calibration method for quantitative Raman measurements on aqueous solutions

    Duraipandian, S., Knopp, Matthias Manne, Pollard, M. R., Kerdoncuff, H., Petersen, J. C. & Mullertz, Anette , 7 Aug 2018, In: Analytical Methods. 10, 29, p. 3589-3593

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Continuous electromembrane extraction coupled with mass spectrometry – Perspectives and challenges

    Fuchs, D., Hidalgo, C. R., Payán, M. D. R., Petersen, Nickolaj J., Jensen, H., Kutter, Jörg P. & Pedersen-Bjergaard, Stig, 2018, In: Analytica Chimica Acta. 999, p. 27-36

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Solid lipid Particles as Drug Carriers - Effects of Particle Preparation Methods and Lipid Excipients on Particle Characteristics

    Gamboa, C. K., Samir, R., Wu, C. & Mu, Huiling, 20 Apr 2018, In: Pharmaceutical Nanotechnology. 6, 2, p. 124-132

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    pH-Triggered nanostructural transformations in antimicrobial peptide/oleic acid self-assemblies

    Gontsarik, M., Mohammadtaheri, M., Yaghmur, Anan & Salentinig, S., 26 Mar 2018, In: Biomaterials Science. 6, 4, p. 803-812 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Bioconjugation of Supramolecular Metallacages to Integrin Ligands for Targeted Delivery of Cisplatin

    Han, J., Räder, A. F. B., Reichart, F., Aikman, B., Wenzel, M. N., Woods, B., Weinmüller, M., Ludwig, B. S., Stürup, Stefan, Groothuis, G. M. M., Permentier, H. P., Bischoff, R., Kessler, H., Horvatovich, P. & Casini, A., 21 Nov 2018, In: Bioconjugate Chemistry. 29, 11, p. 3856-3865 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Manipulating Aggregation Behavior of the Uncharged Peptide Carbetocin

    Høgstedt, U. B., Østergaard, Jesper, Weiss, T., Sjögren, H. & van de Weert, Marco, Mar 2018, In: Journal of Pharmaceutical Sciences. 107, 3, p. 838-847 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Temperature triggering of kinetically trapped self-assemblies in citrem-phospholipid nanoparticles

    Prajapati, R., Salentinig, S. & Yaghmur, Anan, Nov 2018, In: Chemistry and Physics of Lipids. 216, p. 30-38 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Development and validation of an ICP-MS method for quantification of total carbon and platinum in cell samples and comparison of open-vessel and microwave-assisted acid digestion methods

    Riisom, M., Gammelgaard, Bente, Lambert, Ian Henry & Stürup, Stefan, 2018, In: Journal of Pharmaceutical and Biomedical Analysis. 158, p. 144-150 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Structural characterization of self-assemblies of new omega-3 lipids: docosahexaenoic acid and docosapentaenoic acid monoglycerides

    Shao, X., Bor, G., Al-Hosayni, S., Salentinig, S. & Yaghmur, Anan, 7 Oct 2018, In: Physical chemistry chemical physics : PCCP. 20, 37, p. 23928-23941 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Relevance of Copper and Organic Cation Transporters in the Activity and Transport Mechanisms of an Anticancer Cyclometallated Gold(III) Compound in Comparison to Cisplatin

    Spreckelmeyer, S., van der Zee, M., Bertrand, B., Bodio, E., Stürup, Stefan & Casini, A., 2018, In: Frontiers in Chemistry. 6, 15 p., 377.

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Concomitant monitoring of implant formation and drug release of in situ forming poly (lactide-co-glycolide acid) implants in a hydrogel matrix mimicking the subcutis using UV–vis imaging

    Sun, Y., Jensen, H., Petersen, Nickolaj J., Larsen, Susan Weng & Østergaard, Jesper, 2018, In: Journal of Pharmaceutical and Biomedical Analysis. 150, p. 95-106

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    UV-vis Imaging of Piroxicam Supersaturation, Precipitation, and Dissolution in a Flow-Through Setup

    Sun, Y., Chapman, A., Larsen, Susan Weng, Jensen, H., Petersen, Nickolaj J., Goodall, D. M. & Østergaard, Jesper, 5 Jun 2018, In: Analytical Chemistry. 90, 11, p. 6413-6418

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Laser-assisted delivery enhances topical uptake of the anticancer agent cisplatin

    Wenande, E., Olesen, U. H., Boesen, M. R., Persson, Daniel Pergament, Lerche, C. M., Stürup, Stefan, Gammelgaard, Bente, Husted, Søren, Anderson, R. R. & Hædersdal, Merete, 2018, In: Drug Delivery. 25, 1, p. 1877-1885

    Research output: Contribution to journalJournal articleResearchpeer-review

  42. Published

    Effects of a novel selenosugar on primary human vascular cells, mouse aortic rings and atherosclerosis in apoE-/- mice: [Meeting Abstract]

    Zacharias, T., Flouda, K., Jepps, T., Christoffersen, Christina, Pedersen, T., Gammelgaard, Bente, Schiesser, C. & Davies, Michael J., 20 May 2018, In: Free Radical Biology & Medicine. 120, S1, p. S68-S68 P-79.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  43. Published

    UV imaging in pharmaceutical analysis

    Østergaard, Jesper, 5 Jan 2018, In: Journal of Pharmaceutical and Biomedical Analysis. 147, p. 140-148

    Research output: Contribution to journalReviewResearchpeer-review

  44. 2017
  45. Published

    An optimised method for routine separation and quantification of major alkaloids in Cortex Cinchona by HPLC coupled with UV and fluorescence detection.

    Holmfred, Else Skovgaard, Cornett, Claus, Maldonado, C., Rønsted, Nina & Hansen, S. H., Sep 2017, In: Phytochemical Analysis. 28, 5, p. 374-380 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Adjuvants based on synthetic mycobacterial cord factor analogues: Biophysical properties of neat glycolipids and nano-self-assemblies with DDA

    Kallerup, R. S., Franzyk, Henrik, Schiøth, M. L., Justesen, S., Martin-Bertelsen, Birte, Rose, F., Madsen, C. M., Christensen, D., Korsholm, K. S., Yaghmur, Anan & Foged, Camilla, 12 May 2017, In: Molecular Pharmaceutics. 14, 7, p. 2294-2306 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  47. Published

    Phylogeny predicts the quantity of antimalarial alkaloids within the iconic yellow Cinchona bark (Rubiaceae: Cinchona calisaya)

    Maldonado Goyzueta, C. B., Barnes, Christopher James, Cornett, Claus, Holmfred, Else Skovgaard, Hansen, S. H., Persson, C., Antonelli, A. & Rønsted, Nina, 2017, In: Frontiers in Plant Science. 8, 16 p., 391.

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    In Situ Monitoring of Nanostructure Formation during the Digestion of Mayonnaise

    Salentinig, S., Amenitsch, H. & Yaghmur, Anan, 30 Apr 2017, In: ACS Omega. 2, 4, p. 1441-1446 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Mitigating Cyanide Poisoning

    Suman, S. G., Gretarsdottir, J. M., Lambert, Ian Henry & Stürup, Stefan, Jul 2017, p. S261-S261.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  50. 2016
  51. Published

    Taylor Dispersion Analysis as a promising tool for assessment of peptide-peptide interactions

    Høgstedt, U. B., Schwach, G., van de Weert, Marco & Østergaard, Jesper, 25 Jul 2016, In: European Journal of Pharmaceutical Sciences. 93, p. 21-28 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  52. Published

    Delivery of siRNA Complexed with Palmitoylated α-Peptide/β-Peptoid Cell-Penetrating Peptidomimetics: Membrane Interaction and Structural Characterization of a Lipid-Based Nanocarrier System.

    Jing, X., Foged, Camilla, Martin-Bertelsen, Birte, Yaghmur, Anan, Knapp, K. M., Malmsten, M., Franzyk, Henrik & Nielsen, Hanne Mørck, 6 Jun 2016, In: Molecular Pharmaceutics. 13, 6, p. 1739-1749 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  53. Published

    Conserved molecular superlattices in a series of homologous synthetic mycobacterial cell-wall lipids forming interdigitated bilayers

    Martin-Bertelsen, Birte, Yaghmur, Anan, Franzyk, Henrik, Justesen, S., Kirkensgaard, Jacob Judas Kain & Foged, Camilla, 7 Nov 2016, In: Langmuir. 32, 48, p. 12693–12701 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  54. Published

    Nano-self-assemblies based on synthetic analogues of mycobacterial monomycoloyl glycerol and DDA: Supramolecular structure and adjuvant efficacy

    Martin-Bertelsen, Birte, Korsholm, K. S., Christensen, D., Franzyk, Henrik, Yaghmur, Anan & Foged, Camilla, 2016, In: Molecular Pharmaceutics. 13, 8, p. 2771-2781 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review