Sven Frøkjær
Professor, emeritus
- 1996
- Published
Drug delivery studies in Caco-2 monolayers. IV. Ethyl glycoside esters as a novel type of absorption enhancers.
Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1996, In: STP pharma sciences. p. 157-161Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Drug delivery studies in Caco-2 monolayers V. Ethyl glucoside esters as a novel type of absorption enhancers
Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1 Mar 1996, In: S.T.P. Pharma Sciences. 6, 2, p. 157-161 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 1997
- Published
Beta-carboxylic acid esterfied D-Asp-Ala retains a high affinity for the oligopeptide transporter in Caco-2 cell monolayers
Taub, M. E., Larsen, B. D., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 146, p. 205-212 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Influence of oligopeptide transporter binding affinity upon uptake and transport of D-Asp(Obzl)-Ala and Asp(OBzl)-Sar in filter-grown Caco-2 monolayers
Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 156, p. 219-228 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The effect of beta-turn structure on the permeation of peptides across monolayers of bovine brain microvessel endothelial cells
Sørensen, M., Steenberg, B., Knipp, G., Wang, W., Steffansen, B., Frøkjær, Sven & Borchardt, R. T., 1997, In: Pharmaceutical Research. 14, p. 1341-1348Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The novel oxygenated chalcone, 2,4-dimethoxy-4'-butoxychalcone, exhibits potent activity against human malaria parasite Plasmodium falciparum in vitro and rodent parasites Plasmodium berghei and Plasmodium yoelii in vivo
Chen, M., Christensen, Søren Brøgger, Zhai, L., Rasmussen, M. H., Theander, Thor Grundtvig, Frøkjær, Sven, Steffansen, B., Davidsen, J. & Kharazmi, A., 1997, In: Journal of Infectious Diseases. 176, 5, p. 1327-33 6 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 1998
- Published
Assessment of side-chain modified dipeptides that interact with the oligopeptide transporter
Frøkjær, Sven, Steffansen, B. & Taub, M. E., 1998, Peptide and Protein Drug Delivery: Alfred Benzon Symposium 43. Munkgaard, p. 287-297 10 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- Published
Oligopeptide transporter mediated uptake and transport of D-Asp(OBzl)-Ala, D-Glu(OBzl)-Ala and D-Ser(Bzl)-Ala in filter grown Caco-2 monolayers
Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1998, In: International Journal of Pharmaceutics. 174, p. 223-232 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Peptide and protein drug delivery : proceedings of a symposium held at the Royal Danish Academy of Sciences and Letters, August 17-21, 1997: Alfred Benzon Symposium, 43
Frøkjær, Sven, Christrup, Lona Louring, Krogsgaard-Larsen, Povl & Alfred Benzon, F., 1998, Copenhagen: Munksgaard .Research output: Book/Report › Book › Research
- 1999
- Published
Stability metabolism and transport of D-Asp(OBzl)Ala -a model prodrug with affinity for the oligopeptide transporter
Steffansen, B., Lepist, E., Frøkjær, Sven, Taub, M. E. & Lennernas, H., 1999, In: European Journal of Pharmaceutical Sciences. 8, p. 67-73Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Phase behavior and lipid-membrane structure of phospholipid- glycosphingolipid liposomes and the thermal unfolding of insulin
Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 1 Jan 1999, In: Journal of Liposome Research. 9, 2, p. 261-274 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2000
- Published
Stability and vitro metabolism of dipeptide model prodrugs with affinity for the oligopeptide transporter
Lepist, E., Steffansen, B., Kusk, T., Larsen, D. H., Andersen, D., Frøkjær, Sven, Taub, M. E., Veski, P. & Lennernas, H., 2000, In: European Journal of Pharmaceutical Sciences. 11, p. 43-50 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2001
- Published
Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line
Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven, Taub, M. E. & Steffansen, B., 2001, In: Journal of Controlled Release. 76, 1-2, p. 129-38 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line
Nielsen, C. U., Amstrup, J., Steffansen, B., Frøkjær, Sven & Larsen, Birger Brodin, 2001, In: American Journal of Physiology: Gastrointestinal and Liver Physiology. 281, 1, p. G191-9Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Model prodrugs for the intestinal oligopeptide transporter: model drug release in aqueous solution and in various biological media
Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2001, In: Journal of Controlled Release. 73, 1, p. 21-30 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Enzymatic degradation of polymer covered SOPC-liposomes in relation to drug delivery
Davidsen, Johan, Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 29 Jan 2001, In: Advances in Colloid and Interface Science. 89-90, p. 303-311 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Association of an acylated model peptide with DPPC-DPPS lipid membranes
Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 77-81 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Drug delivery by phospholipase A2 degradable liposomes
Davidsen, J., Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 67-69 3 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Association of acylated cationic decapeptides with dipalmitoylphosphatidylserine-dipalmitoylphosphatidylcholine lipid membranes
Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 7 Nov 2001, In: Chemistry and Physics of Lipids. 113, 1-2, p. 83-95 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2002
- Published
Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line
Nielsen, C. U., Supuran, C. T., Scozzafava, A., Frøkjær, Sven, Steffansen, B. & Larsen, Birger Brodin, 2002, In: Pharmaceutical Research. 19, 9, p. 1337-44 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1
Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B. & Frøkjær, Sven, 2002, In: Basic & Clinical Pharmacology & Toxicology. 90, 6, p. 285-96 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A calorimetric study of phosphocholine membranes mixed with desmopressin and its diacylated prodrug derivative (DPP)
Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 21 Feb 2002, In: International Journal of Pharmaceutics. 233, 1-2, p. 199-206 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Human peptide transporters: Therapeutic applications
Nielsen, C. U., Larsen, Birger Brodin, Jørgensen, Flemming Steen, Frøkjær, Sven & Steffansen, B., 1 Sep 2002, In: Expert Opinion on Therapeutic Patents. 12, 9, p. 1329-1350 22 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2003
- Published
Prodrugs
Steffansen, B., Thomsen, A. E. & Frøkjær, Sven, 2003, Estimation of solubility, permeability, absorption and bioavaibility. van de Waterbeemd, H., Lennernäs, H. & Artursson, P. (eds.). Weinheim: Wiley-VCH, p. 532-546Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research
- Published
Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism
Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 2003, In: Journal of Controlled Release. 86, 2-3, p. 279-92 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1298692
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Risk Perceptions in Diabetic Patients Who Have Experienced Adverse Events: Implications for Patient Involvement in Regulatory Decisions
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Guidance for pediatric use in prescription information for novel medicinal products in the EU and the US
Research output: Contribution to journal › Journal article › Research › peer-review
Published