Birger Brodin Larsen
Professor
CNS Drug Delivery and Barrier Modelling
Universitetsparken 2
2100 København Ø
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miRNA-27a-3p and miRNA-222-3p as Novel Modulators of Phosphodiesterase 3a (PDE3A) in Cerebral Microvascular Endothelial Cells
Yasmeen, S., Kaur, S., Mirza, A. H., Larsen, Birger Brodin, Pociot, Flemming & Kruuse, Christina Rostrup, Aug 2019, In: Molecular Neurobiology. 56, 8, p. 5304–5314Research output: Contribution to journal › Journal article › Research › peer-review
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mRNA expression and transport function of the proton-coupled amino acid transporter, PAT1, along the rat intestine
Broberg, M. L., Larsen, K. B., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., 2010.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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mRNA expression and transport function of the proton-coupled amino acid transporter , PAT1, along the rat intestine
Broberg, M. L., Brandt Larsen, K., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., Mar 2010. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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iP-gp , a novel cell line with tight barrier function and expression of human P-glycoprotein (ABCB1) for drug screening
Larsen, Birger Brodin, Ozgür, Burak & Saaby, Lasse, 23 May 2017.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3
Søndergaard, H. B., Larsen, Birger Brodin & Nielsen, C. U., 2008, In: Pflügers Archiv: European Journal of Physiology. 456, 3, p. 611-622Research output: Contribution to journal › Journal article › Research › peer-review
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hPEPT1 Affinity and Translocation of Selected Gln-Sar and Glu-Sar Dipeptide Derivatives
Eriksson, A. H., Elm, P. L., Begtrup, M., Nielsen, R., Steffansen, B. & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 3, p. 242-249Research output: Contribution to journal › Journal article › Research › peer-review
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d-Aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1)
Frølund, S., Marquez, O. C., Larsen, M., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 159, 6, p. 1339-1353Research output: Contribution to journal › Journal article › Research › peer-review
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Vigabatrin absorption is mediated via the proton-coupled amino acid transporter PAT1 – in vitro and in vivo
Nøhr, M. K., Juul, R. V., Hansen, S. H., Larsen, Birger Brodin, Holm, R., Kreilgaard, M. & Nielsen, C. U., 24 Jun 2013.Research output: Contribution to conference › Poster › Research
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Validation of reference genes for normalization of real-time quantitative PCR studies of gene expression in brain capillary endothelial cells cultured in vitro
Hersom, M., Goldeman, C., Pretzer, N. & Larsen, Birger Brodin, Dec 2018, In: Molecular and Cellular Neuroscience. 93, p. 27-35 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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VPS10P domain receptor trafficking in brain endothelial cells
Siupka, P., Højland, A., Thomsen, L. B., Lykke-Hartmann, K., Helms, H. C. C., Larsen, Birger Brodin, Moos, T., Madsen, P. S. & Nielsen, M. S., 10 Dec 2014. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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Two-photon fluorescence imaging: a platform to investigate cell-penetrating peptides and liposome-based nanocarriers for drug delivery across the heterogeneous BBB in vivo
Kucharz, K., Kristensen, K., Kristensen, Mie, Lund, M., Andresen, T., Larsen, Birger Brodin & Lauritzen, M., 2019, In: Journal of Cerebral Blood Flow and Metabolism. 39, p. 60 1 p.Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
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Transport pathways mediating blood-to-brain L-glutamate efflux
Helms, H. C. C., Nielsen, C. U., Waagepetersen, Helle S. & Larsen, Birger Brodin, 10 Dec 2014. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1
Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B. & Frøkjær, Sven, 2002, In: Basic & Clinical Pharmacology & Toxicology. 90, 6, p. 285-96 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Transport of amino acids and GABA analogues via the human proton-coupled amino acid transporter, hPAT1: Characterization of conditions for affinity and transport experiments in Caco-2 cells.
Larsen, M., Larsen, Birger Brodin, Frølund, Bente & Nielsen, C. U., 2008, In: European Journal of Pharmaceutical Sciences. 35, 1-2, p. 86-95Research output: Contribution to journal › Journal article › Research › peer-review
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Transport of Gaboxadol via hPAT1 and rOAT1 in the absence and presence of 5-HTP
Broberg, M. L., Holm, R., Larsen, Birger Brodin, Jensen, K. G. & Nielsen, C. U., 29 Jul 2009. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line
Nielsen, C. U., Supuran, C. T., Scozzafava, A., Frøkjær, Sven, Steffansen, B. & Larsen, Birger Brodin, 2002, In: Pharmaceutical Research. 19, 9, p. 1337-44 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Transport af lægemiddelstoffer gennem vævsbarrier
Nielsen, C. U. & Larsen, Birger Brodin, 2011, Bioteknologi - en temabog. Gasbjerg, P. K., Jensen, G. S. & Sørensen, A. B. (eds.). Århus: Systime, p. 145-157 12 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Education › peer-review
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Transferrin receptor expression and role in transendothelial transport of transferrin in cultured brain endothelial monolayers
Hersom, M., Helms, H. C., Pretzer, N., Andersen, C. G., Jensen, A. I., Severin, G., Nielsen, M. S., Holm, R. & Larsen, Birger Brodin, 24 Aug 2016, In: Molecular and Cellular Neuroscience. 76, p. 59-67 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Transendothelial electrical resistance measurement across the blood–brain barrier: A critical review of methods
Vigh, J. P., Kincses, A., Ozgür, Burak, Walter, F. R., Santa-Maria, A. R., Valkai, S., Vastag, M., Neuhaus, W., Larsen, Birger Brodin, Dér, A. & Deli, M. A., 2021, In: Micromachines. 12, 6, 18 p., 685.Research output: Contribution to journal › Review › Research › peer-review
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The putative P-gp inhibitor telmisartan does not affect the transcellular permeability and cellular uptake of the calcium channel antagonist verapamil in the P-glycoprotein expressing cell line MDCK II MDR1
Saaby, Lasse, Tfelt-Hansen, P. & Larsen, Birger Brodin, 11 Jun 2015, In: Pharmacology Research & Perspectives. 3, 4, p. 1-9 9 p., e00151.Research output: Contribution to journal › Journal article › Research › peer-review
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The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics
Frølund, S., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 161, 3, p. 589-600Research output: Contribution to journal › Journal article › Research › peer-review
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The proton-coupled amino acid transporter hPAT1 is the main transporter involved in vigabatrin uptake in intestinal Caco-2 cells
Nøhr, M. K., Hansen, S. H., Larsen, Birger Brodin, Holm, R. & Nielsen, C. U., 30 Nov 2012.Research output: Contribution to conference › Poster › Research
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The interaction of CNS-active Amaryllidae alkaloids with the BBB efflux pump MDR1
Eriksson, A. H., Birrer, A., Sendra, J. R., Güler, S., Rønsted, Nina, Jäger, A. K. & Larsen, Birger Brodin, 29 Jun 2010. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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The insulin receptor is expressed and functional in cultured blood-brain barrier endothelial cells, but does not mediate insulin entry from blood-to-brain
Hersom, M., Helms, H. C., Schmalz, C., Pedersen, T. Å., Buckley, S. T. & Larsen, Birger Brodin, 2018, In: American Journal of Physiology: Endocrinology and Metabolism. 315, 4, p. E531-E542Research output: Contribution to journal › Journal article › Research › peer-review
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The insulin receptor is expressed and functional in blood-brain barrier endothelial cells, but does not mediate insulin entry from blood-to-brain
Hersom, M. N. S., Helms, H. C. C., Pedersen, T., Buckley, S. & Larsen, Birger Brodin, 14 Sep 2016.Research output: Contribution to conference › Conference abstract for conference › Research
ID: 1299175
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Design of prodrugs targeting the intestinal di/tri‐peptide transporter hPEPT1 (SLC15A1
Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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233
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A bovine in vitro blood-brain barrier model under oxygenglucose deprivation (OGD) condition
Research output: Contribution to conference › Poster › Research
Published