Drug Delivery and Biophysics of Biopharmaceuticals

  1. Published

    Inhalable siRNA-loaded nano-embedded microparticles engineered using microfluidics and spray drying

    Agnoletti, M., Bohr, A., Thanki, K., Wan, F., Zeng, X., Bøtker, Johan Peter, Yang, Mingshi & Foged, Camilla, Nov 2017, In: European Journal of Pharmaceutics and Biopharmaceutics. 120, p. 9-21

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Monosized Polymeric Microspheres Designed for Passive Lung Targeting: Biodistribution and Pharmacokinetics after Intravenous Administration

    Agnoletti, M., Rodríguez-Rodríguez, C., Klodzinska, S. N., Esposito, T., Saatchi, K., Nielsen, Hanne Mørck & Häfeli, U. O., 2020, In: ACS Nano. 14, p. 6693-6706

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Peptide-Membrane Interactions Monitored by Fluorescence Lifetime Imaging: A Study Case of Transportan 10

    Anselmo, S., Sancataldo, G., Nielsen, Hanne Mørck, Foderà, Vito & Vetri, V., 2021, In: Langmuir. 37, 44, p. 13148-13159

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    α-casein micelles-membranes interaction: Flower-like lipid protein coaggregates formation

    Anselmo, S., Sancataldo, G., Foderà, Vito & Vetri, V., 2022, In: Biochimica et Biophysica Acta - General Subjects. 1866, 10, 11 p., 130196.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Sustainable soy protein microsponges for efficient removal of lead (II) from aqueous environments

    Anselmo, S., Avola, T., Kalouta, Kleopatra, Cataldo, S., Sancataldo, G., Muratore, N., Foderà, Vito, Vetri, V. & Pettignano, A., 2023, In: International Journal of Biological Macromolecules. 239, 14 p., 124276.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Impact of drug loading in mesoporous silica-amorphous formulations on the physical stability of drugs with high recrystallization tendency

    Antonino, R. S. C. M. Q., Ruggiero, M., Song, Z., Nascimento, T. L., Lima, E. M., Bohr, A., Knopp, Matthias Manne & Löbmann, Korbinian, 2019, In: International Journal of Pharmaceutics: X. 1, 7 p., 100026.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Models to predict intestinal absorption of therapeutic peptides and proteins

    Antunes, F., Andrade, F., Ferreira, D., Nielsen, Hanne Mørck & Sarmento, B., Jan 2013, In: Current Drug Metabolism. 14, 1, p. 4-20 17 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Cell-Penetrating Peptides as Tools to Facilitate Oral Delivery of Biopharmaceuticals

    Asgreen, Camilla Jantzen, Fredholt, Freja, Nielsen, Hanne Mørck & Kristensen, Mie, 2023, Cell-Penetrating Peptides: Design, Development and Applications. Oba, M. & Demizu, Y. (eds.). Wiley-VCH, p. 331-354

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  9. Published

    Cell-penetrating antimicrobial peptides - prospectives for targeting intracellular infections

    Bahnsen, J. S., Franzyk, Henrik, Sayers, E. J., Jones, A. T. & Nielsen, Hanne Mørck, 2015, In: Pharmaceutical Research. 32, 5, p. 1546-56 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Repurposing azithromycin and rifampicin against Gram-negative pathogens by combination with peptide potentiators

    Baker, K. R., Jana, B., Hansen, A. M., Vissing, K. J., Nielsen, Hanne Mørck, Franzyk, Henrik & Guardabassi, Luca, 2019, In: International Journal of Antimicrobial Agents. 53, p. 868-872 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Repurposing Azithromycin and Rifampicin Against Gram-Negative Pathogens by Combination With Peptidomimetics

    Baker, K. R., Jana, B., Hansen, A. M., Nielsen, Hanne Mørck, Franzyk, Henrik & Guardabassi, Luca, 2 Jul 2019, In: Frontiers in Cellular and Infection Microbiology. 9

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Fluorophore labeling of a cell-penetrating peptide induces differential effects on its cellular distribution and affects cell viability

    Birch, D., Christensen, M. V., Stærk, Dan, Franzyk, Henrik & Nielsen, Hanne Mørck, 2017, In: B B A - Biomembranes. 1859, 12, p. 2483-2494

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Stereoisomer-Dependent Membrane Association and Capacity for Insulin Delivery Facilitated by Penetratin

    Birch, D., Sayers, E. J., Christensen, M. V., Jones, A. T., Franzyk, Henrik & Nielsen, Hanne Mørck, 2023, In: Pharmaceutics. 15, 6, 15 p., 1672.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Evaluation of drug permeation under fed state conditions using mucus-covered Caco-2 cell epithelium

    Birch, D., Diedrichsen, Ragna Guldsmed, Christophersen, P. C., Mu, Huiling & Nielsen, Hanne Mørck, Jun 2018, In: European Journal of Pharmaceutical Sciences. 118, p. 144-153

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Stereochemistry as a determining factor for the effect of a cell-penetrating peptide on cellular viability and epithelial integrity

    Birch, D., Christensen, M. V., Stærk, Dan, Franzyk, Henrik & Nielsen, Hanne Mørck, 24 May 2018, In: Biochemical Journal. 475, 10, p. 1773-1788 16 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Comparative study of the drug delivery mechanism of L-penetratin and D-penetratin

    Birch, D., Christensen, M. V., Stærk, Dan, Franzyk, Henrik & Nielsen, Hanne Mørck, 2018.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  17. Published

    Direct observations of drug nanocarrier interactions and mobility within biological interfaces

    Bohr, S. S. R., Streck, S., Pinholt, H., Wan, F., Mcdowell, A., Nielsen, Hanne Mørck & Hatzakis, Nikos, 2022, In: Biophysical Journal. 121, 3, p. 72a-73a 2 p., 355-Pos.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  18. Published

    Quantitative Evaluation of a Multimodal Aptamer-Targeted Long-Circulating Polymer for Tumor Targeting

    Bohrmann, L., Burghardt, T., Rodríguez-Rodríguez, C., Herth, Matthias Manfred, Saatchi, K. & Häfeli, U. O., 2023, In: ACS Omega. 8, 12, p. 11003-11020

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Aptamers used for molecular imaging and theranostics: recent developments

    Bohrmann, L., Burghardt, T., Haynes, C., Saatchi, K. & Häfeli, U. O., 2022, In: Theranostics. 12, 9, p. 4010-4050

    Research output: Contribution to journalReviewResearchpeer-review

  20. Published

    Interaction with prefibrillar species and amyloid-like fibrils changes the stiffness of lipid bilayers

    Borro, B. C., Parolini, L., Cicuta, P., Foderà, Vito & Di Michele, L., 25 Oct 2017, In: Physical chemistry chemical physics : PCCP. 19, 41, p. 27930-27934 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    On the purported "backbone fluorescence" in protein three-dimensional fluorescence spectra

    Bortolotti, A., Wong, Y. H., Korsholm, S. S., Bahring, N. H. B., Bobone, S., Tayyab, S., van de Weert, Marco & Stella, L., 2016, In: RSC Advances. 6, 114, p. 112870-112876 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Amphiphilic-DNA Platform for the Design of Crystalline Frameworks with Programmable Structure and Functionality

    Brady, R. A., Brooks, N. J., Foderà, Vito, Cicuta, P. & Di Michele, L., 14 Nov 2018, In: Journal of the American Chemical Society. 140, 45, p. 15384-15392

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Flexibility defines structure in crystals of amphiphilic DNA nanostars

    Brady, R. A., Kaufhold, W. T., Brooks, N. J., Foderà, Vito & Di Michele, L., 2019, In: Journal of Physics: Condensed Matter. 31, 7, 11 p., 0704003.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Drug delivery studies in Caco-2 monolayers. III. Intestinal transport of various vasopressin analogues in the presence of lysophosphatidylcholine

    Brøndsted, H., Nielsen, Hanne Mørck & Hovgaard, L., 14 Feb 1995, In: International Journal of Pharmaceutics. 114, 2, p. 151-157 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Disentangling the role of solvent polarity and protein solvation in folding and self-assembly of α-lactalbumin

    Bucciarelli, S., Sayedi, E. S., Osella, S., Trzaskowski, B., Vissing, K. J., Vestergaard, Bente & Foderà, Vito, 2020, In: Journal of Colloid and Interface Science. 561, p. 749-761 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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