Research areas

  1. Published

    Affinity and translocation relationships via hPEPT1 of H-Xaa-Ser-OH dipeptides: evaluation of H-Phe-Ser-OH as a pro-moiety for ibuprofen and benzoic acid prodrugs

    Omkvist, D. H., Trangbæk, D. J., Mildon, J., Paine, J. S., Larsen, Birger Brodin, Begtrup, M. & Nielsen, C. U., 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 77, 2, p. 327-331

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1)

    Omkvist, D. H., Larsen, S. B., Nielsen, C. U., Steffansen, B., Olsen, L., Jørgensen, Flemming Steen & Larsen, Birger Brodin, 2010, In: The AAPS Journal. 12, 3, p. 385-396

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 161, 8, p. 1793-1805

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010.

    Research output: Contribution to conferencePosterResearch

  5. Published

    Intestinal drug delivery via hPEPT1 : in vitro and in silico evaluation of the realtionship between substrate, binding and translocation

    Omkvist, D. H., Feb 2011, Det Farmaceutiske Fakultet. 51 p.

    Research output: Book/ReportPh.D. thesisResearch

  6. Published

    Constituents in kava extracts potentially involved in hepatotoxicity: A review

    Olsen, L. R., Grillo, M. P. & Skonberg, C., 2011, In: Chemical Research in Toxicology. 24, p. 992-1002

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Prediction of activation energies for hydrogen abstraction by cytochrome p450

    Olsen, L., Rydberg, P., Rod, T. H. & Ryde, U., 2006, In: Journal of Medicinal Chemistry. 49, 22, p. 6489-6499

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Hvad har varme at gøre med lægemidler?

    Olsen, L., Kasper, C., Kastrup, Jette Sandholm Jensen, Gajhede, Michael & Jørgensen, Flemming Steen, 2006, In: Lægemiddelforskning. p. 31-33

    Research output: Contribution to journalJournal articleCommunication

  9. Published

    Cytochrome P450 Mediated Drug Metabolism

    Olsen, L., Jørgensen, Flemming Steen & Oostenbrink, C., 2016, New Horizons in Predictive Drug Metabolism and Pharmacokinetics. Wilson, A. G. E. (ed.). Cambridge: Royal Society of Chemistry, p. 66-78 13 p. (RSC Drug Discovery, Vol. 49).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  10. Published

    Determination of leukocyte DNA 6-thioguanine nucleotide levels by high-performance liquid chromatography with fluorescence detection

    Olsen, K., Hansen, S. H., Sidenius, U. & Schmiegelow, Kjeld, 2008, In: Journal of Chromatography - B. 864, 1-2, p. 149-155

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Studies on the metabolism of tolmetin to the chemically reactive acyl-coenzyme a thioester intermediate in rats

    Olsen, J., Li, C., Skonberg, C., Bjørnsdottir, I., Sidenius, U., Benet, L. Z. & Hansen, S. H., 2007, In: Drug Metabolism and Disposition. 35, 5, p. 758-764

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Toltrazuril and its two main metabolites in the environment - Analytical development

    Olsen, J., Hansen, M., Krogh, K. A., Bak, S. A., Brandt, A. & Björklund, E., 2011.

    Research output: Contribution to conferencePosterResearch

  13. Published

    Isolation of the MAO-inhibitor naringenin from Mentha aquatica L

    Olsen, H. T., Stafford, G. I., van Staden, J., Christensen, Søren Brøgger & Jäger, A. K., 2008, In: Journal of Ethnopharmacology. 117, 3, p. 500-502

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Peptoid-Peptide hybrid backbone architectures

    Olsen, Christian Adam, 25 Jan 2010, In: ChemBioChem. 11, 2, p. 152-160

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Antimicrobial, hemolytic, and cytotoxic activities of ß-peptoid-peptide hybrid oligomers: Improved properties compared to natural AMPs

    Olsen, Christian Adam, Ziegler, H. L., Nielsen, Hanne Mørck, Frimodt-Møller, N., Jaroszewski, J. W. & Franzyk, Henrik, 2010, In: ChemBioChem. 11, 10, p. 1356-1360

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Small molecules from spiders used as chemical probes

    Olsen, C. A., Kristensen, Anders Skov & Strømgaard, Kristian, 25 Nov 2011, In: Angewandte Chemie International Edition. 50, 48, p. 11296-11311

    Research output: Contribution to journalReviewResearchpeer-review

  17. Published

    Solid-phase synthesis of neuroactive spider-wasp hybrid toxin analogues using a backbone amide linker

    Olsen, Christian Adam, Witt, M., Franzyk, Henrik & Jaroszewski, J. W., 2007, In: Tetrahedron Letters. 48, 3, p. 405-408

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Aziridines in parallel- and solid-phase synthesis

    Olsen, Christian Adam, Bonke, G., Vedel, L., Franzyk, Henrik & Jaroszewski, J. W., 2007, In: European Journal of Organic Chemistry. 2007, 11, p. 1717-1724

    Research output: Contribution to journalReviewResearchpeer-review

  19. Published

    Solid-phase peptide synthesis and circular dichroism study of chiral ß-peptoid homooligomers

    Olsen, Christian Adam, Lambert, M., Witt, M., Franzyk, Henrik & Jaroszewski, J. W., 2008, In: Amino Acids. 34, 3, p. 465-471

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    α-Peptide/ß-Peptoid Chimeras

    Olsen, Christian Adam, Bonke, G., Vedel, L., Adsersen, A., Witt, M., Franzyk, Henrik & Jaroszewski, J. W., 2007, In: Organic Letters. 9, 8, p. 1549–1552 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Hyraceum, the fossilized metabolic product of rock hyraxes (Procavia capensis), shows GABA-benzodiazepine receptor affinity

    Olsen, A., Prinsloo, L. C., Scott, L. & Jäger, A. K., 2008, In: South African Journal of Science. 103, 11/12, p. 437-438

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Translational pain research: evaluating analgesic effect in experimental visceral pain models

    Olesen, A. E., Andresen, T., Christrup, Lona Louring & Upton, R. N., 2009, In: World Journal of Gastroenterology. 15, 2, p. 177-81

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Forskelle på ordinationsmønstret af analgetika ved behandling af cancersmerter på seks danske smertebehandlingsenheder

    Olesen, A. E., Jarvig, L., Hansen, O. B., Højsted, J., von Holstein-Rathlou, Niels-Henrik, Jonsson, T., Sjøgren, P., Sonne, N. M., Sørensen, J. T. & Christrup, Lona Louring, 2007, In: Ugeskrift for læger. 169, 21, p. 2024-9

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    A pharmacokinetic and pharmacodynamic study of oral oxycodone in a human experimental pain model of hyperalgesia

    Olesen, A. E., Upton, R., Staahl, C., Christrup, Lona Louring, Arendt-Nielsen, L. & Drewes, A. M., 2010, In: Clinical Pharmacokinetics. 49, 12, p. 817-827

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    The use of biorelevant dissolution media in determining the region of microemulsion: Implications for in vitro lipid formulation assessment

    Ogbonna, A., Ren, S., Olesen, P. & Mullertz, Anette , 2009.

    Research output: Contribution to conferencePosterResearch

  26. Published

    From consumerism to active dependence: patterns of medicines use and treatment decisions among patients with atopic dermatitis

    Nørreslet, M., Bissell, P. & Traulsen, Janine Marie, 2010, In: Health. 14, 1, p. 91-106

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Real-time monitoring of the progerss of polymerization reactions directly on surfaces at open atmosphere by ambient mass spectrometry

    Nørgaard, A. W., Vaz, B. G., Lauritsen, F. R. & Eberlin, M. N., 2010, In: Rapid Communications in Mass Spectrometry. 24, p. 3441-3446

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Characterization of nanofilm spray products by mass spectrometry

    Nørgaard, A. W., Wolkoff, P. & Lauritsen, F. R., 2010, In: Chemosphere. 80, p. 1377-1386

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Nebulization ionization and desorption ionization analysis of reactive organofunctionalized silanes in nanofilm products

    Nørgaard, A. W., Janfelt, Christian, Benassi, M., Wolkoff, P. & Lauritsen, F. R., 2011, In: Journal of Mass Spectrometry. 46, 4, p. 402-410

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    The antagonistic effect of antipsychotic drugs on a HEK293 cell line stably expressing human alpha(1A1)-adrenoceptors

    Nourian, Z., Mulvany, M. J., Nielsen, K. B., Pickering, Darryl S & Kristensen, T., 2008, In: European Journal of Pharmacology. 596, 1-3, p. 32-40

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Critical evaluation of the FANTOM3 non-coding RNA transcripts

    Nordström, K. J. V., Mirza, M. A. I., Almén, M. S., Gloriam, David E., Fredriksson, R. & Schiöth, H. B., 2009, In: Genomics. 94, 3, p. 169-176

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Immunity by formulation design: induction of high CD8+ T-cell responses by poly (I:C) incorporated into the CAF01 adjuvant via a double emulsion method

    Nordly, P. J., Rose, F., Christensen, D., Nielsen, Hanne Mørck, Andersen, P., Agger, E. M. & Foged, Camilla, 2011, In: Journal of Controlled Release. 150, 3, p. 307-317

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Innovativt nanopartikeldesign bag skræddersyede vacciner

    Nordly, P. J., Agger, E. M., Nielsen, Hanne Mørck & Foged, Camilla, 2009, In: Lægemiddelforskning. p. 19-21

    Research output: Contribution to journalJournal articleResearch

  34. Published

    Incorporation of the TLR4 agonist monophosphoryl lipid A into the bilayer of DDA/DTDB liposomes : physico-chemical characterization and induction of CD8+ T-Cell responses in vivo

    Nordly, P. J., Agger, E. M., Andersen, P., Nielsen, Hanne Mørck & Foged, Camilla, 2011, In: Pharmaceutical Research. 28, 3, p. 553-562

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Formulation of vaccine adjuvants: modulating the adjuvant activity of DDA/TDB liposomes with immunopotentiators

    Nordly, P. J., 2010, København: Det Farmaceutiske Fakultet.

    Research output: Book/ReportPh.D. thesisResearch

  36. Published

    Status and future prospects of lipid-based particulate delivery systems as vaccine adjuvants and their combination with immunostimulators

    Nordly, P. J., Madsen, H. B., Nielsen, Hanne Mørck & Foged, Camilla, 2009, In: Expert Opinion on Drug Delivery. 6, 7, p. 1-16

    Research output: Contribution to journalReviewResearch

  37. Published

    A synthetic mycobacterial monomycoloyl glycerol analogue stabilizes DDA liposomes

    Nordly, P. J., Pedersen, E. A., Khiljii, T. S., Agger, E. M., Jørgensen, Lene, Nielsen, Hanne Mørck, Korsholm, K. S., Franzyk, Henrik & Foged, Camilla, 2010, In: CRS Newsletter. 27, 2, p. 12 14 p.

    Research output: Contribution to journalJournal articleResearch

  38. Published

    Incorporation of a synthetic mycobacterial monomycoloyl glycerol analogue stabilizes dimethyldioctadecylammonium liposomes and potentiates their adjuvant effect in vivo

    Nordly, P. J., Korsholm, K. S., Pedersen, E. A., Khilji, T. S., Franzyk, Henrik, Jørgensen, Lene, Nielsen, Hanne Mørck, Agger, E. M. & Foged, Camilla, 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 77, 1, p. 89-98

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Drying of firewood - the effect of harvesting time, tree species and shelter of stacked wood

    Nord-Larsen, Thomas, Bergstedt, A. C. E., Farver, O. & Heding, Niels, 2011, In: Biomass & Bioenergy. 35, 7, p. 2993-2998 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Application of Q2MM to stereoselective reactions

    Nilsson Lill, S. O., Forbes, A., Donoghue, P., Verdolino, V., Wiest, O., Rydberg, P. & Norrby, P., Sep 2010, In: Current Organic Chemistry. 14, 15, p. 1629-1645

    Research output: Contribution to journalReviewResearchpeer-review

  41. Published

    Triazoloquinazolinediones as novel high affinity ligands for the benzodiazepine site of GABA(A) receptors

    Nilsson, J., Gidlöf, R., Nielsen, E. Ø., Liljefors, T., Nielsen, M. P. C. & Sterner, O., 1 Jan 2011, In: Bioorganic & Medicinal Chemistry. 19, 1, p. 111-121

    Research output: Contribution to journalJournal articleResearchpeer-review

  42. Published

    3-Alkyl- and 3-amido-isothiazoloquinolin-4-ones as ligands for the benzodiazepine site of GABAA receptors

    Nilsson, J., Nielsen, E. Ø., Liljefors, T., Nielsen, M. P. C. & Sterner, O., Feb 2012, In: Bioorganic Chemistry. 40, p. 125-130

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABAA receptors

    Nilsson, J., Nielsen, E. Ø., Liljefors, T., Nielsen, M. P. C. & Sterner, O., 2008, In: Bioorganic & Medicinal Chemistry Letters. 18, 21, p. 5713-5716

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Positive modulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors reverses subcronic PCP-induced deficits in the novel object recognition task in rats

    Nielsen, T. D., Larsen, D. B., Hansen, S. L., Grayson, B., Neill, J. C. & Plath, N., 11 Feb 2010, In: Behavioural Brain Research. 207, 1, p. 144-150 7 p.

    Research output: Contribution to journalJournal articleResearch

  45. Published

    Investigation of the mnemonic deficits in the sub-chronic PCP model of schizophrenia

    Nielsen, T. D., 2010, København: Museum Tusculanum. 73 p.

    Research output: Book/ReportPh.D. thesisResearch

  46. Published

    Determination of protein conformation by isotopically labelled cross-linking and dedicated software: Application to the chaperone, calreticulin

    Nielsen, T., Thaysen-Andersen, M., Larsen, N., Jørgensen, Flemming Steen, Houen, G. & Højrup, P., 2007, In: International Journal of Mass Spectrometry. 268, 2-3, p. 217-226

    Research output: Contribution to journalJournal articleResearchpeer-review

  47. Published

    Topics in mathematical modelling, K.K. Tung. Princeton University Press (2007). 300 pages

    Nielsen, S. N., 2008, In: Ecological Modelling. 211, 1-2, p. 247-248

    Research output: Contribution to journalLiterature reviewResearch

  48. Published

    Towards an ecosystem semiotics. Some basic aspects for a new research programme

    Nielsen, S. N., 2007, In: Ecological Complexity : An International Journal on Biocomplexity in the Environment and Theoretical Ecology. 4, 3, p. 93-101

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Ny bog til biofagenes videnskabsteori

    Nielsen, S. N., 2007, In: MONA: Matematik og Naturfagsdidaktik. 1, p. 71-74

    Research output: Contribution to journalLiterature reviewResearch

  50. Published

    Understanding the functional principles of nature - proposing another type of ecosystem services

    Nielsen, S. N. & Müller, F., 2009, In: Ecological Modelling. 220, p. 1913-1925

    Research output: Contribution to journalJournal articleResearchpeer-review

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