Sven Frøkjær

Sven Frøkjær

Professor, emeritus


  1. 2022
  2. Published

    Guidance for pediatric use in prescription information for novel medicinal products in the EU and the US

    Christiansen, H., De Bruin, M. L., Frøkjær, Sven & Hallgreen, Christine Erikstrup, 2022, In: PLoS ONE. 17, 4, 19 p., e0266353.

    Research output: Contribution to journalJournal articlepeer-review

  3. 2020
  4. Published

    Data-enriched edible pharmaceuticals (DEEP) of medical cannabis by inkjet printing

    Öblom, H., Cornett, Claus, Bøtker, Johan Peter, Frøkjær, Sven, Hansen, Harald S., Rades, Thomas, Rantanen, Jukka & Genina, Natalja, 2020, In: International Journal of Pharmaceutics. 589, p. 1-11 119866.

    Research output: Contribution to journalJournal articlepeer-review

  5. 2019
  6. Published

    Danish Physicians’ Views on the Appropriateness of the Involvement of Patients with Type 2 Diabetes in Regulatory Decision Making: A Qualitative Study

    Sachs, M. L., Colding-Jørgensen, M., Helboe, P., Kälvemark Sporrong, Sofia, Frøkjær, Sven, Jelic, K. & Kaae, Susanne, 2019, In: Pharmaceutical Medicine. 33, 2, p. 99-107

    Research output: Contribution to journalJournal articlepeer-review

  7. 2017
  8. Published

    Risk Perceptions in Diabetic Patients Who Have Experienced Adverse Events: Implications for Patient Involvement in Regulatory Decisions

    Sachs, M. L., Kälvemark Sporrong, Sofia, Colding-Jørgensen, M., Frøkjær, Sven, Helboe, P., Jelic, K. & Kaae, Susanne, 2017, In: Pharmaceutical Medicine. 31, 4, p. 245-255 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  9. 2015
  10. Published

    Den danske kodeks for integritet i forskning

    Pedersen, H. M., Frøkjær, Sven, Bach, L. W., Vestergaard, E., Pedersen, C. V., Dirckinck-Holmfeld, L., Wegener, H. C., Jensen, L., Staunstrup, J. & Hansen, J. M., 2015

    Research output: Book/ReportReport

  11. 2013
  12. Published

    Medicon Valley - dansk-svensk succes

    Jørgensen, S., Ahren, B., Jensen, I. S. & Frøkjær, Sven, 14 Mar 2013, In: Morgenavisen Jyllands-Posten. p. 28

    Research output: Contribution to journalContribution to newspaper - Feature article

  13. Published

    Biologiske lægemidler - fra molekyle til medicin

    Nielsen, Hanne Mørck, Foged, Camilla, Jørgensen, Lene & Frøkjær, Sven, 2013, In: Lægemiddelforskning. p. 12-14

    Research output: Contribution to journalJournal article

  14. Published

    Influence of acylation on the adsorption of GLP-2 to hydrophobic surfaces

    Pinholt, C., Kapp, S. J., Bukrinsky, J. T., Hostrup, S., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2013, In: International Journal of Pharmaceutics. 440, 1, p. 63-71 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  15. 2012
  16. Published

    Calcipotriol delivery into the skin with PEGylated liposomes

    Knudsen, N. Ø., Rønholt, Stine, Salte, R. D., Jørgensen, Lene, Thormann, T., Basse, L. H., Hansen, J., Frøkjær, Sven & Foged, Camilla, 2012, In: European Journal of Pharmaceutics and Biopharmaceutics. 81, 3, p. 532-9 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  17. Published

    Design of cyclic RKKH peptide-conjugated PEG liposomes targeting the integrin a2ß1 receptor

    Knudsen, N. Ø., Schiffelers, R. M., Jørgensen, Lene, Hansen, J., Frøkjær, Sven & Foged, Camilla, 2012, In: International Journal of Pharmaceutics. 428, 1-2, p. 171-177

    Research output: Contribution to journalJournal articlepeer-review

  18. 2011
  19. Published

    Influence of PEGylation with linear and branched PEG chains on the adsorption of glucagon to hydrophobic surfaces

    Pinholt, C., Bukrinsky, J. T., Hostrup, S., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 77, 1, p. 139-147

    Research output: Contribution to journalJournal articlepeer-review

  20. Published

    Influence of acylation on the adsorption of insulin to hydrophobic surfaces

    Pinholt, C., Hostrup, S., Bukrinsky, J. T., Frøkjær, Sven & Jørgensen, Lene, 2011, In: Pharmaceutical Research. 28, p. 1031-1040

    Research output: Contribution to journalJournal articlepeer-review

  21. Published

    Ionic strength-dependent denaturation of Thermomyces lanuginosus lipase induced by SDS

    Fanø, M., van de Weert, Marco, Møller, E. H., Kruse, N. A. & Frøkjær, Sven, 2011, In: Archives of Biochemistry and Biophysics. 506, 1, p. 92-98

    Research output: Contribution to journalJournal articlepeer-review

  22. Published

    Targeting of liposome-associated calcipotriol to the skin: effect of liposomal membrane fluidity and skin barrier integrity

    Knudsen, N. Ø., Jørgensen, Lene, Hansen, J., Vermehren, C., Frøkjær, Sven & Foged, Camilla, 2011, In: International Journal of Pharmaceutics. 416, p. 478-485

    Research output: Contribution to journalJournal articlepeer-review

  23. 2010
  24. Published

    Influence of glycosylation on the adsorption of Thermomyces lannuginosus lipase to hydrophobic and hydrophilic surfaces

    Pinholt, C., Fanø, M., Wiberg, C., Hostrup, S., Bukrinsky, J. T., Frøkjær, Sven, Norde, W. & Jørgensen, Lene, 2010, In: European Journal of Pharmaceutical Sciences. 40, 4, p. 273-281

    Research output: Contribution to journalJournal articlepeer-review

  25. Published

    Issues in Development of Biodrug Delivery Systems

    Jørgensen, Lene, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, Biodrug Delivery Systems: Fundamentals, Applications and Clinical Development. Morishita, M. & Park, K. (eds.). 1 ed. Informa Healthcare, p. 13-25

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  26. Published

    Issues in development of biodrug delivery systems

    Jørgensen, Lene, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, Biodrug delivery systems: fundamentals, applications and clinical development. Morishita, M. & Park, K. (eds.). New York: Informa Healthcare, p. 13-25

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  27. Published

    Penetration of gel and liquid state liposomes into barrier-impaired skin

    Knudsen, N. Ø., Frøkjær, Sven, Hansen, J., Jørgensen, Lene & Foged, Camilla, 2010, In: Journal of Pharmacy and Pharmacology. p. 793

    Research output: Contribution to journalConference articlepeer-review

  28. Published

    Preparation and characterization of poly (DL-lactide-co-glycolide) nanoparticles for siRNA delivery

    Cun, D., Foged, Camilla, Yang, Mingshi, Frøkjær, Sven & Nielsen, Hanne Mørck, 2010, In: Internation Journal of Pharmaceutics. 390, 1, p. 70-75

    Research output: Contribution to journalJournal articlepeer-review

  29. Published

    Spray drying of siRNA-containing PLGA nanoparticles intended for inhalation

    Jensen, D. M. K., Cun, D., Maltesen, M. J., Frøkjær, Sven, Nielsen, Hanne Mørck & Foged, Camilla, 2010, In: Journal of Controlled Release. 142, p. 138-145

    Research output: Contribution to journalJournal articlepeer-review

  30. 2009
  31. Published

    Biotechnology-based pharmaceuticals

    Jørgensen, Lene, Nielsen, Hanne Mørck & Frøkjær, Sven, 2009, Modern pharmaceutics: applications and advances. Florence, A. T. & Siepmann, J. (eds.). 5 ed. New York: Informa Healthcare, Vol. 2. p. 259-293 (Drugs and the Pharmaceutical Sciences, Vol. 188).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  32. Published

    Formation mechanism of insulin fibrils and structural aspects of the insulin fibrillation process

    Jensen, M. G., Frøkjær, Sven & Vestergaard, Bente, 2009, In: Current Protein and Peptide Science. 10, 5, p. 509-528

    Research output: Contribution to journalJournal articlepeer-review

  33. Published

    Novel formulation approaches for peptide and protein injectables

    Yang, Mingshi & Frøkjær, Sven, 2009, Delivery technologies for biopharmaceuticals: Peptides, proteins, nucleic acids and vaccines. Jørgensen, L. & Mørck Nielsen, H. (eds.). Wiley, p. 11-28

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  34. 2008
  35. Published

    Cellular uptake and membrane-destabilising properties of a-peptide/ß-peptoid chimeras: lessons for the design of new cell-penetrating peptides

    Foged, Camilla, Franzyk, Henrik, Bahrami, S., Frøkjær, Sven, Jaroszewski, J. W., Nielsen, Hanne Mørck & Olsen, Christian Adam, 2008, In: BBA General Subjects. 1778, 11, p. 2487-2495

    Research output: Contribution to journalJournal articlepeer-review

  36. Published

    Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1

    Søndergaard, H. B., Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2008, In: European Journal of Pharmaceutical Sciences. 33, 4-5, p. 332-342

    Research output: Contribution to journalJournal articlepeer-review

  37. Published

    Metode til screening af modificerede proteinlægemidler under opbevaring

    Petersen, C., Jørgensen, Lene, Hostrup, S., Bukrinsky, J. T. & Frøkjær, Sven, 2008, In: Lægemiddelforskning. p. 16-18

    Research output: Contribution to journalJournal article

  38. 2007
  39. Published

    A helical structural nucleus is the primary elongating unit of insulin amyloid fibrils

    Vestergaard, Bente, Jensen, M. G., Roessle, M., Kastrup, Jette Sandholm Jensen, van de Weert, Marco, Flink, J. M., Frøkjær, Sven, Gajhede, Michael & Svergun, D. I., 2007, In: PLoS - Biology. 5, 5, p. 1089-1097

    Research output: Contribution to journalJournal articlepeer-review

  40. Published

    Binding mode of Thioflavin T in insulin amyloid fibrils

    Jensen, M. G., Norrman, M., Flink, J. M., van de Weert, Marco, Bukrinsky, J. T., Schluckebier, G. & Frøkjær, Sven, 2007, In: Journal of Structural Biology. 159, 3, p. 483-497

    Research output: Contribution to journalJournal articlepeer-review

  41. Published

    Characterisation and physical stability of PEGylated glucagon

    Stigsnæs, P., Frøkjær, Sven, Bjerregaard, S., van de Weert, Marco, Kingshott, P. & Møller, E. H., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 89-98

    Research output: Contribution to journalJournal articlepeer-review

  42. Published

    Characterisation of salmon calcitonin in spray-dried powder for inhalation. Effect of chitosan

    Yang, Mingshi, Velaga, S., Yamamoto, H., Takeuchi, H., Kawashima, Y., Hovgaard, L., van de Weert, Marco & Frøkjær, Sven, 2007, In: Internation Journal of Pharmaceutics. 331, 2, p. 176-181

    Research output: Contribution to journalJournal articlepeer-review

  43. Published

    Computational prediction of solubilizers' effect on partitioning

    Høst, J., Christensen, I. T., Jørgensen, Flemming Steen, Frøkjær, Sven & Hovgaard, L., 2007, In: Internation Journal of Pharmaceutics. 329, 1-2, p. 46-52

    Research output: Contribution to journalJournal articlepeer-review

  44. Published

    Gennembrud i forståelsen af insulinfibrillering

    Jensen, M. G., Vestergaard, Bente, Frøkjær, Sven, Gajhede, Michael, Flink, J. M., van de Weert, Marco, Kastrup, Jette Sandholm Jensen & Svergun, D. I., 2007, In: Lægemiddelforskning. p. 10-11

    Research output: Contribution to journalJournal article

  45. Published

    I-125 used for labelling of proteins in an absorption model changes the absorption rate of insulin aspart

    Søhoel, A., Plum, A., Frøkjær, Sven & Thygesen, P., 2007, In: Internation Journal of Pharmaceutics. 330, 1-2, p. 114-120

    Research output: Contribution to journalJournal articlepeer-review

  46. Published

    Liposomes for phospholipase A2 triggered siRNA release: preparation and in vitro test

    Foged, Camilla, Nielsen, Hanne Mørck & Frøkjær, Sven, 2007, In: Internation Journal of Pharmaceutics. 331, 2, p. 160-166

    Research output: Contribution to journalJournal articlepeer-review

  47. Published

    Phospholipase A2 sensitive liposomes for delivery of small interfering RNA (siRNA)

    Foged, Camilla, Nielsen, Hanne Mørck & Frøkjær, Sven, 2007, In: Journal of Liposome Research. 17, 3-4

    Research output: Contribution to journalJournal articlepeer-review

  48. Published

    Study on the binding of Thioflavin T to ß-sheet-rich and non-ß-sheet cavities

    Jensen, M. G., Olsen, L., van de Weert, Marco, Flink, J. M., Frøkjær, Sven & Jørgensen, Flemming Steen, 2007, In: Journal of Structural Biology. 158, 3, p. 358-369

    Research output: Contribution to journalJournal articlepeer-review

  49. 2006
  50. Published

    Chemical and thermal stability of insulin: effects of zinc and ligand binding to the insulin zinc-hexamer

    Huus, K., Havelund, S., Olsen, H. B., van de Weert, Marco & Frøkjær, Sven, Nov 2006, In: Pharmaceutical Research. 23, 11, p. 2611-20 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  51. Published

    Ligand binding and thermostability of different allosteric states of the insulin zinc-hexamer

    Huus, K., Havelund, S., Olsen, H. B., Sigurskjold, B. W., van de Weert, Marco & Frøkjær, Sven, 28 Mar 2006, In: Biochemistry. 45, 12, p. 4014-4024 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  52. Published

    Kinetics of insulin adsorption at the oil-water interface and diffusion properties of adsorbed layers monitored using fluorescence correlation spectroscopy

    Donsmark, J., Jørgensen, Lene, Mollmann, S., Frøkjær, Sven & Rischel, C., 1 Jan 2006, In: Pharmaceutical Research. 23, 1, p. 148-155 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  53. Published

    In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1

    Andersen, R., Nielsen, C. U., Begtrup, M., Jørgensen, Flemming Steen, Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2006, In: European Journal of Pharmaceutical Sciences. 28, 4, p. 325-35 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  54. Published

    Interfacial adsorption of insulin - conformational changes and reversibility of adsorption

    Mollmann, S. H., Jørgensen, Lene, Bukrinsky, J. T., Elofsson, U., Norde, W. & Frøkjær, Sven, 2006, In: European Journal of Pharmaceutical Sciences. 27, 2-3, p. 194-204

    Research output: Contribution to journalJournal articlepeer-review

  55. Published

    Kinetics of insulin adsorption and gelation at the oil-water interface monitored using fluorescence correlation spectroscopy

    Donsmark, J., Jørgensen, Lene, Mollmann, S. H., Frøkjær, Sven & Rischel, C., 2006, In: Pharmaceutical Research. 23, 1, p. 148-155

    Research output: Contribution to journalJournal articlepeer-review

  56. Published

    Preparing and evaluating delivery systems for proteins

    Jorgensen, L., Moeller, E. H., van de Weert, Marco, Nielsen, H. M. & Frøkjær, Sven, 2006, In: European Journal of Pharmaceutical Sciences. 29, 3-4, p. 174-82 9 p.

    Research output: Contribution to journalReviewpeer-review

  57. 2005
  58. Published

    Factors of importance for a successful delivery system for proteins

    van de Weert, Marco, Jørgensen, Lene, Horn Moeller, E. & Frøkjær, Sven, Nov 2005, In: Expert Opinion on Drug Delivery. 2, 6, p. 1029-37 9 p.

    Research output: Contribution to journalReviewpeer-review

  59. Published

    Phase behavior and nanoscale structure of phospholipid membranes incorporated with acylated C14-peptides

    Pedersen, T. B., Kaasgaard, T., Jensen, M., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., Oct 2005, In: Biophysical Journal. 89, 4, p. 2494-2503 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  60. Published

    Thermal dissociation and unfolding of insulin

    Huus, K., Havelund, S., Olsen, H. B., van de Weert, Marco & Frøkjær, Sven, 23 Aug 2005, In: Biochemistry. 44, 33, p. 11171-7 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  61. Published

    Complex coacervation with heparin results in decreased lysozyme stability

    van de Weert, Marco, Bendix Andersen, M. & Frøkjær, Sven, 3 Jan 2005, In: Journal of controlled release : official journal of the Controlled Release Society. 101, 1-3, p. 361-2 2 p.

    Research output: Contribution to journalConference abstract in journal

  62. Published

    Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media

    Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 2, p. 98-108 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  63. Published

    Delivery aspects of small peptides and substrates for peptide transporters

    Steffansen, B., Nielsen, C. U. & Frøkjær, Sven, 2005, In: European Journal of Pharmaceutics and Biopharmaceutics. 60, 4, p. 241-245 4 p.

    Research output: Contribution to journalReviewpeer-review

  64. Published

    Evaluation of statistical design/modeling for prediction of the effect of amino acids on agitation-induced aggregation of human growth hormone and human insulin

    Soenderkaer, S., van de Weert, Marco, Lindgaard Hansen, L., Flink, J. & Frøkjær, Sven, 2005, In: Journal of Drug Delivery Science and Technology. 15, 6, p. 427-434 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  65. Published

    Particle size and surface charge affect particle uptake by human dendritic cells in an in vitro model

    Foged, Camilla, Larsen, Birger Brodin, Frøkjær, Sven & Sundblad, A., 2005, In: Internation Journal of Pharmaceutics. 298, 2, p. 315-22 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  66. 2004
  67. Published

    Complex coacervation of lysozyme and heparin: complex characterization and protein stability

    van de Weert, Marco, Andersen, M. B. & Frøkjær, Sven, Dec 2004, In: Pharmaceutical Research. 21, 12, p. 2354-9 6 p.

    Research output: Contribution to journalJournal articlepeer-review

  68. Published

    Probing structural changes of proteins incorporated into water-in-oil emulsions

    Jørgensen, Lene, van de Weert, Marco, Vermehren, C., Bjerregaard, S. & Frøkjær, Sven, Jul 2004, In: Journal of Pharmaceutical Sciences. 93, 7, p. 1847-59 13 p.

    Research output: Contribution to journalJournal articlepeer-review

  69. Published

    Effects of sucrose on rFVIIa aggregation and methionine oxidation

    Soenderkaer, S., Carpenter, J. F., van de Weert, Marco, Hansen, L. L., Flink, J. & Frøkjær, Sven, Apr 2004, In: European Journal of Pharmaceutical Sciences. 21, 5, p. 597-606 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  70. Published

    In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model

    Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 1 Jan 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 77-86 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  71. Published

    Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2

    Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 2004, In: American Journal of Physiology - Renal Physiology. 286, 2, p. 385-393

    Research output: Contribution to journalJournal articlepeer-review

  72. Published

    Formulation, stability and characterization of protein and peptide drugs

    Frøkjær, Sven, Hovgaard, L. & van de Weert, Marco, 2004, Biomaterials for Delivery and Targeting of Proteins and Nucleic Acids. Mahato, R. I. (ed.). Boca Raton: CRC Press, p. 378-401

    Research output: Chapter in Book/Report/Conference proceedingBook chapterCommunication

  73. Published

    In vitro release of insulin aspart incorporated into water-in-oil emulsions

    Jørgensen, Lene, Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2004, In: Journal of Drug Delivery Science and Technology. 14, 6, p. 455-459

    Research output: Contribution to journalJournal articlepeer-review

  74. Published

    Interaction of dendritic cells with antigen-containing liposomes: effect of bilayer composition

    Foged, Camilla, Arigita, C., Sundblad, A., Jiskoot, W., Storm, G. & Frøkjær, Sven, 2004, In: Vaccine. 22, 15-16, p. 1903-13 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  75. Published

    Intestinal solute carriers: an overview of trends and strategies for improving oral drug absorption

    Steffansen, B., Nielsen, C. U., Larsen, Birger Brodin, Eriksson, A. H., Andersen, R. & Frøkjær, Sven, 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 3-16 14 p.

    Research output: Contribution to journalJournal articlepeer-review

  76. Published

    Micropipette manipulation a technique to evaluate the stability of water-in-oil emulsions containing proteins

    Jørgensen, Lene, Kim, D. H., Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2004, In: Journal of Pharmaceutical Sciences. 93, 12, p. 2994-3003

    Research output: Contribution to journalJournal articlepeer-review

  77. 2003
  78. Published

    In vitro and in vivo aspects of N-acyl-phosphatidylethanolamine-containing liposomes

    Vermehren, Charlotte, Clausen-Beck, B., Frøkjær, Sven & Hansen, Harald S., 18 Mar 2003, In: International Journal of Pharmaceutics. 254, 1, p. 49-53 5 p.

    Research output: Contribution to journalJournal articlepeer-review

  79. Published

    Erratum: Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: Affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism (Journal of Controlled Release (2003) 86 (279-292) PII: S0168365902004133)

    Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 7 Mar 2003, In: Journal of Controlled Release. 88, 2

    Research output: Contribution to journalJournal articlepeer-review

  80. Published

    Prodrugs

    Steffansen, B., Thomsen, A. E. & Frøkjær, Sven, 2003, Estimation of solubility, permeability, absorption and bioavaibility. van de Waterbeemd, H., Lennernäs, H. & Artursson, P. (eds.). Weinheim: Wiley-VCH, p. 532-546

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  81. Published

    Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism

    Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 2003, In: Journal of Controlled Release. 86, 2-3, p. 279-92 14 p.

    Research output: Contribution to journalJournal articlepeer-review

  82. Published

    Secondary structure alteration in insulin and growth hormone water-in-oil emulsions

    Jørgensen, Lene, Vermehren, Charlotte, Bjerregaard, S. & Frøkjær, Sven, 2003, In: Internation Journal of Pharmaceutics. 254, 1, p. 7-10

    Research output: Contribution to journalJournal articlepeer-review

  83. 2002
  84. Published

    Human peptide transporters: Therapeutic applications

    Nielsen, C. U., Larsen, Birger Brodin, Jørgensen, Flemming Steen, Frøkjær, Sven & Steffansen, B., 1 Sep 2002, In: Expert Opinion on Therapeutic Patents. 12, 9, p. 1329-1350 22 p.

    Research output: Contribution to journalJournal articlepeer-review

  85. Published

    A calorimetric study of phosphocholine membranes mixed with desmopressin and its diacylated prodrug derivative (DPP)

    Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 21 Feb 2002, In: International Journal of Pharmaceutics. 233, 1-2, p. 199-206 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  86. Published

    Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line

    Nielsen, C. U., Supuran, C. T., Scozzafava, A., Frøkjær, Sven, Steffansen, B. & Larsen, Birger Brodin, 2002, In: Pharmaceutical Research. 19, 9, p. 1337-44 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  87. Published

    Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1

    Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B. & Frøkjær, Sven, 2002, In: Basic & Clinical Pharmacology & Toxicology. 90, 6, p. 285-96 12 p.

    Research output: Contribution to journalJournal articlepeer-review

  88. 2001
  89. Published

    Association of acylated cationic decapeptides with dipalmitoylphosphatidylserine-dipalmitoylphosphatidylcholine lipid membranes

    Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 7 Nov 2001, In: Chemistry and Physics of Lipids. 113, 1-2, p. 83-95 13 p.

    Research output: Contribution to journalJournal articlepeer-review

  90. Published

    Association of an acylated model peptide with DPPC-DPPS lipid membranes

    Pedersen, T. B., Sabra, M. C., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 77-81 5 p.

    Research output: Contribution to journalJournal articlepeer-review

  91. Published

    Drug delivery by phospholipase A2 degradable liposomes

    Davidsen, J., Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 19 Feb 2001, In: International Journal of Pharmaceutics. 214, 1-2, p. 67-69 3 p.

    Research output: Contribution to journalJournal articlepeer-review

  92. Published

    Enzymatic degradation of polymer covered SOPC-liposomes in relation to drug delivery

    Davidsen, Johan, Vermehren, Charlotte, Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 29 Jan 2001, In: Advances in Colloid and Interface Science. 89-90, p. 303-311 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  93. Published

    Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line

    Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven, Taub, M. E. & Steffansen, B., 2001, In: Journal of Controlled Release. 76, 1-2, p. 129-38 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  94. Published

    Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line

    Nielsen, C. U., Amstrup, J., Steffansen, B., Frøkjær, Sven & Larsen, Birger Brodin, 2001, In: American Journal of Physiology: Gastrointestinal and Liver Physiology. 281, 1, p. G191-9

    Research output: Contribution to journalJournal articlepeer-review

  95. Published

    Model prodrugs for the intestinal oligopeptide transporter: model drug release in aqueous solution and in various biological media

    Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2001, In: Journal of Controlled Release. 73, 1, p. 21-30 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  96. 2000
  97. Published

    Stability and vitro metabolism of dipeptide model prodrugs with affinity for the oligopeptide transporter

    Lepist, E., Steffansen, B., Kusk, T., Larsen, D. H., Andersen, D., Frøkjær, Sven, Taub, M. E., Veski, P. & Lennernas, H., 2000, In: European Journal of Pharmaceutical Sciences. 11, p. 43-50 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  98. 1999
  99. Published

    Phase behavior and lipid-membrane structure of phospholipid- glycosphingolipid liposomes and the thermal unfolding of insulin

    Pedersen, T. B., Frøkjær, Sven, Mouritsen, Ole G. & Jørgensen, K., 1 Jan 1999, In: Journal of Liposome Research. 9, 2, p. 261-274 14 p.

    Research output: Contribution to journalJournal articlepeer-review

  100. Published

    Stability metabolism and transport of D-Asp(OBzl)Ala -a model prodrug with affinity for the oligopeptide transporter

    Steffansen, B., Lepist, E., Frøkjær, Sven, Taub, M. E. & Lennernas, H., 1999, In: European Journal of Pharmaceutical Sciences. 8, p. 67-73

    Research output: Contribution to journalJournal articlepeer-review

  101. 1998
  102. Published

    Assessment of side-chain modified dipeptides that interact with the oligopeptide transporter

    Frøkjær, Sven, Steffansen, B. & Taub, M. E., 1998, Peptide and Protein Drug Delivery: Alfred Benzon Symposium 43. Munkgaard, p. 287-297 10 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  103. Published

    Oligopeptide transporter mediated uptake and transport of D-Asp(OBzl)-Ala, D-Glu(OBzl)-Ala and D-Ser(Bzl)-Ala in filter grown Caco-2 monolayers

    Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1998, In: International Journal of Pharmaceutics. 174, p. 223-232 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  104. Published
  105. 1997
  106. Published

    Beta-carboxylic acid esterfied D-Asp-Ala retains a high affinity for the oligopeptide transporter in Caco-2 cell monolayers

    Taub, M. E., Larsen, B. D., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 146, p. 205-212 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  107. Published

    Influence of oligopeptide transporter binding affinity upon uptake and transport of D-Asp(Obzl)-Ala and Asp(OBzl)-Sar in filter-grown Caco-2 monolayers

    Taub, M. E., Moss, B. A., Steffansen, B. & Frøkjær, Sven, 1997, In: International Journal of Pharmaceutics. 156, p. 219-228 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  108. Published

    The effect of beta-turn structure on the permeation of peptides across monolayers of bovine brain microvessel endothelial cells

    Sørensen, M., Steenberg, B., Knipp, G., Wang, W., Steffansen, B., Frøkjær, Sven & Borchardt, R. T., 1997, In: Pharmaceutical Research. 14, p. 1341-1348

    Research output: Contribution to journalJournal articlepeer-review

  109. Published

    The novel oxygenated chalcone, 2,4-dimethoxy-4'-butoxychalcone, exhibits potent activity against human malaria parasite Plasmodium falciparum in vitro and rodent parasites Plasmodium berghei and Plasmodium yoelii in vivo

    Chen, M., Christensen, Søren Brøgger, Zhai, L., Rasmussen, M. H., Theander, Thor Grundtvig, Frøkjær, Sven, Steffansen, B., Davidsen, J. & Kharazmi, A., 1997, In: Journal of Infectious Diseases. 176, 5, p. 1327-33 6 p.

    Research output: Contribution to journalJournal articlepeer-review

  110. 1996
  111. Published

    Drug delivery studies in Caco-2 monolayers V. Ethyl glucoside esters as a novel type of absorption enhancers

    Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1 Mar 1996, In: S.T.P. Pharma Sciences. 6, 2, p. 157-161 5 p.

    Research output: Contribution to journalJournal articlepeer-review

  112. Published

    Drug delivery studies in Caco-2 monolayers. IV. Ethyl glycoside esters as a novel type of absorption enhancers.

    Nielsen, Hanne Mørck, Brøndsted, H., Frøkjær, Sven & Hovgaard, L., 1996, In: STP pharma sciences. p. 157-161

    Research output: Contribution to journalJournal articlepeer-review

ID: 1298692