Korbinian Löbmann

Korbinian Löbmann

Guest Researcher


  1. 2024
  2. Published

    Analysis of stabilization mechanisms in β-lactoglobulin-based amorphous solid dispersions by experimental and computational approaches

    Zhuo, Xuezhi, Foderà, Vito, Larsson, P., Schaal, Z., Bergström, C. A. S., Löbmann, Korbinian & Kabedev, A., 2024, In: European Journal of Pharmaceutical Sciences. 192, 13 p., 106639.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Effect of Drug Loading in Mesoporous Silica on Amorphous Stability and Performance

    Bavnhøj, C. G., Knopp, Matthias Manne & Löbmann, Korbinian, 2024, In: Pharmaceutics. 16, 2, 11 p., 163.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Exploring the effect of protein secondary structure on the solid state and physical stability of protein-based amorphous solid dispersions

    Zhuo, Xuezhi, Ochner, J., Leng, D., Foderà, Vito & Löbmann, Korbinian, 2024, In: European Journal of Pharmaceutics and Biopharmaceutics. 198, 8 p., 114274.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Investigating the influence of protein secondary structure on the dissolution behavior of β-lactoglobulin-based amorphous solid dispersions

    Zhuo, Xuezhi, Tozzetti, M., Arnous, A., Leng, D., Foderà, Vito & Löbmann, Korbinian, 2024, In: International Journal of Pharmaceutics. 653, 8 p., 123887.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Use of solid thermolytic salts to facilitate microwave-induced in situ amorphization

    Qiang, W., Zhang, M., Löbmann, Korbinian, McCoy, C. P., Andrews, G. P. & Zhao, M., 2024, In: International Journal of Pharmaceutics. 651, 11 p., 123791.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. 2023
  8. Published

    A Comparative Study between A Protein Based Amorphous Formulation and Other Dissolution Rate Enhancing Approaches: A Case Study with Rifaximin

    Zhuo, Xuezhi, Margrethe Brekstad Kjellin, M., Schaal, Z., Zhang, T., Löbmann, Korbinian & Leng, D., 2023, In: Pharmaceutics. 15, 1, 10 p., 126.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Mechanisms of Drug Solubility Enhancement Induced by β-Lactoglobulin-Based Amorphous Solid Dispersions

    Zhuo, Xuezhi, Sener, Z., Kabedev, A., Zhao, M., Arnous, A., Leng, D., Foderà, Vito & Löbmann, Korbinian, 2023, In: Molecular Pharmaceutics. 20, 10, p. 5206–5213

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    The effects of surfactants on the performance of polymer-based microwave-induced in situ amorphization

    Qiang, W., Löbmann, Korbinian, McCoy, C. P., Andrews, G. P. & Zhao, M., 2023, In: International Journal of Pharmaceutics. 630, 17 p., 122426.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. 2022
  12. Published

    Development of a multiparticulate drug delivery system for in situ amorphisation

    Holm, T. P., Kokott, M., Knopp, Matthias Manne, Boyd, Ben, Berthelsen, R., Quodbach, J. & Löbmann, Korbinian, 2022, In: European Journal of Pharmaceutics and Biopharmaceutics. 180, p. 170-180

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Hyperthermia-Induced In Situ Drug Amorphization by Superparamagnetic Nanoparticles in Oral Dosage Forms

    Ansari, S. R., Hempel, N. J., Asad, S., Svedlindh, P., Bergström, C. A. S., Löbmann, Korbinian & Teleki, A., 2022, In: ACS Applied Materials and Interfaces. 14, 19, p. 21978–21988

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Stabilizing Mechanisms of β-Lactoglobulin in Amorphous Solid Dispersions of Indomethacin

    Kabedev, A., Zhuo, Xuezhi, Leng, D., Foderà, Vito, Zhao, M., Larsson, P., Bergström, C. A. S. & Löbmann, Korbinian, 2022, In: Molecular Pharmaceutics. 19, 11, p. 3922–3933

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Supersaturated amorphous solid dispersions of celecoxib prepared in situ by microwave irradiation

    Holm, T. P., Knopp, Matthias Manne, Berthelsen, R. & Löbmann, Korbinian, 2022, In: International Journal of Pharmaceutics. 626, 8 p., 122115.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. 2021
  17. Published

    The effect of the molecular weight of polyvinylpyrrolidone and the model drug on laser-induced in situ amorphization

    Hempel, N. J., Merkl, P., Knopp, Matthias Manne, Berthelsen, R., Teleki, A., Hansen, A. K., Sotiriou, G. A. & Löbmann, Korbinian, Jul 2021, In: Molecules. 26, 13, 13 p., 4035.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published
  19. Published

    Comparison of co-former performance in co-amorphous formulations: Single amino acids, amino acid physical mixtures, amino acid salts and dipeptides as co-formers

    Wu, W., Grohganz, Holger, Rades, Thomas & Löbmann, Korbinian, 2021, In: European Journal of Pharmaceutical Sciences. 156, 8 p., 105582.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Deliquescence Behavior of Deep Eutectic Solvents

    Palmelund, H., Rantanen, Jukka & Löbmann, Korbinian, 2021, In: Applied Sciences. 11, 9 p., 1601.

    Research output: Contribution to journalLetterResearchpeer-review

  21. Published

    Enabling formulations of aprepitant: in vitro and in vivo comparison of nanocrystalline, amorphous and deep eutectic solvent based formulations

    Palmelund, H., Eriksen, J. B., Bauer-Brandl, A., Rantanen, Jukka & Löbmann, Korbinian, 2021, In: International Journal of Pharmaceutics: X. 3, 100083.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Investigation into the role of the polymer in enhancing microwave-induced in situ amorphization

    Qiang, W., Löbmann, Korbinian, Knopp, Matthias Manne, McCoy, C. P., Andrews, G. P. & Zhao, M., 2021, In: International Journal of Pharmaceutics. 609, 8 p., 121157.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Microwave induced in situ amorphisation facilitated by crystalline hydrates

    Holm, T. P., Knopp, M. M., Löbmann, Korbinian & Berthelsen, R., 2021, In: European Journal of Pharmaceutical Sciences. 163, 9 p., 105858.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Microwave-Induced in Situ Drug Amorphization Using a Mixture of Polyethylene Glycol and Polyvinylpyrrolidone

    Hempel, N. J., Knopp, Matthias Manne, Zeitler, J. A., Berthelsen, R. & Löbmann, Korbinian, 2021, In: Journal of Pharmaceutical Sciences. 110, 9, p. 3221-3229

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Predictive identification of co-formers in co-amorphous systems

    Chambers, L. I., Grohganz, Holger, Palmelund, H., Löbmann, Korbinian, Rades, Thomas, Musa, O. M. & Steed, J. W., 2021, In: European Journal of Pharmaceutical Sciences. 157, 9 p., 105636.

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Studying the impact of the temperature and sorbed water during microwave-induced In Situ amorphization: A case study of celecoxib and polyvinylpyrrolidone

    Hempel, N. J., Knopp, Matthias Manne, Löbmann, Korbinian & Berthelsen, R., 2021, In: Pharmaceutics. 13, 6, 13 p., 886.

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    The Influence of Drug-Polymer Solubility on Laser-Induced In Situ Drug Amorphization Using Photothermal Plasmonic Nanoparticles

    Hempel, N., Merkl, P., Knopp, Matthias Manne, Berthelsen, R., Teleki, A., Sotiriou, G. A. & Löbmann, Korbinian, 2021, In: Pharmaceutics. 13, 6, 12 p., 917.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    The Influence of Temperature and Viscosity of Polyethylene Glycol on the Rate of Microwave-Induced In Situ Amorphization of Celecoxib

    Hempel, N., Dao, T., Knopp, Matthias Manne, Berthelsen, R. & Löbmann, Korbinian, 2021, In: Molecules. 26, 1, 8 p., 110.

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    The Use of Glycerol as an Enabling Excipient for Microwave-Induced In Situ Drug Amorphization

    Hempel, N., Morsch, F., Knopp, Matthias Manne, Berthelsen, R. & Löbmann, Korbinian, 2021, In: Journal of Pharmaceutical Sciences. 110, 1, p. 155-163 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Utilizing Laser Activation of Photothermal Plasmonic Nanoparticles to Induce On-Demand Drug Amorphization inside a Tablet

    Hempel, N. J., Merkl, P., Asad, S., Knopp, M. M., Berthelsen, R., Bergström, C. A. S., Teleki, A., Sotiriou, G. A. & Löbmann, Korbinian, 2021, In: Molecular Pharmaceutics. 18, 6, p. 2254–2262

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. 2020
  32. Published

    The influence of drug and polymer particle size on the in situ amorphization using microwave irradiation

    Hempel, N. J., Knopp, Matthias Manne, Berthelsen, R., Zeitler, J. A. & Löbmann, Korbinian, Apr 2020, In: European Journal of Pharmaceutics and Biopharmaceutics. 149, p. 77-84 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Amorphous drug stabilization using mesoporous materials

    Veloso, D. F. M. C., Knopp, Matthias Manne & Löbmann, Korbinian, 2020, Drug delivery trends. Elsevier, Vol. 3. p. 151-166

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  34. Published

    Constraints on CaCO3 precipitation in superabsorbent polymer by aerobic bacteria

    Nielsen, S. D., Koren, K., Löbmann, Korbinian, Hinge, M., Scoma, A., Kjeldsen, K. U. & Roy, H., 2020, In: Applied Microbiology and Biotechnology. 104, 1, p. 365-375

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Convection-Induced vs. Microwave Radiation-Induced in situ Drug Amorphization

    Hempel, N., Knopp, Matthias Manne, Berthelsen, R. & Löbmann, Korbinian, 2020, In: Molecules. 25, 5, 7 p., 1068.

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Formulation of co-amorphous systems from naproxen and naproxen sodium and in situ monitoring of physicochemical state changes during dissolution testing by Raman spectroscopy

    Ueda, H., Bøtker, Johan Peter, Edinger, M., Löbmann, Korbinian, Grohganz, Holger, Mullertz, Anette , Rades, Thomas & Østergaard, Jesper, 2020, In: International Journal of Pharmaceutics. 587, 119662.

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Hot Melt Coating of Amorphous Carvedilol

    Bannow, J., Koren, L., Salar-Behzadi, S., Löbmann, Korbinian, Zimmer, A. & Rades, Thomas, 2020, In: Pharmaceutics. 12, 6, 13 p., 519.

    Research output: Contribution to journalJournal articleResearchpeer-review

  38. Published

    Improving the drug load and in vitro performance of supersaturated self-nanoemulsifying drug delivery systems (super-SNEDDS) using polymeric precipitation inhibitors

    Bannow, J., Yorulmaz, Y., Löbmann, Korbinian, Mullertz, Anette & Rades, Thomas, 2020, In: International Journal of Pharmaceutics. 575, 1188960.

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Influence of the Polymer Glass Transition Temperature and Molecular Weight on Drug Amorphization Kinetics Using Ball Milling

    Asgreen, Camilla Jantzen, Knopp, Matthias Manne, Skytte, J. & Löbmann, Korbinian, 2020, In: Pharmaceutics. 12, 6, 6 p., 483.

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Influence of water of crystallization on the ternary phase behavior of a drug and deep eutectic solvent

    Palmelund, H., Boyd, B. J., Rantanen, Jukka & Löbmann, Korbinian, 2020, In: Journal of Molecular Liquids. 315, p. 1-7 113727.

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Microwave-Induced In Situ Amorphization: A New Strategy for Tackling the Stability Issue of Amorphous Solid Dispersions

    Qiang, W., Löbmann, Korbinian, McCoy, C. P., Andrews, G. P. & Zhao, M., 2020, In: Pharmaceutics. 12, 7, 19 p., 655.

    Research output: Contribution to journalReviewResearchpeer-review

  42. 2019
  43. Published

    The role interplay between mesoporous silica pore volume and surface area and their effect on drug loading capacity

    Bavnhøj, C. G., Knopp, Matthias Manne, Madsen, C. & Löbmann, Korbinian, 1 Dec 2019, In: International Journal of Pharmaceutics: X. 1, 5 p., 100008.

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Direct Measurement of Amorphous Solubility

    Stukelj, J., Svanback, S., Agopov, M., Löbmann, Korbinian, Strachan, C. J., Rades, Thomas & Yliruusi, J., 4 Jun 2019, In: Analytical Chemistry. 91, 11, p. 7411-7417

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    In situ co-amorphisation in coated tablets – The combination of carvedilol with aspartic acid during immersion in an acidic medium

    Petry, I., Löbmann, Korbinian, Grohganz, Holger, Rades, Thomas & Leopold, C. S., 10 Mar 2019, In: International Journal of Pharmaceutics. 558, p. 357-366 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Design of Inhalable Solid Dosage Forms of Budesonide and Theophylline for Pulmonary Combination Therapy

    Leng, D., Kissi, E. O., Löbmann, Korbinian, Thanki, K., Fattal, E., Rades, Thomas, Foged, Camilla & Yang, Mingshi, 7 Mar 2019, In: AAPS PharmSciTech. 20, 3, 137.

    Research output: Contribution to journalJournal articleResearchpeer-review

  47. Published

    Transformations between Co-Amorphous and Co-Crystal Systems and Their Influence on the Formation and Physical Stability of Co-Amorphous Systems

    Wu, W., Wang, Y., Löbmann, Korbinian, Grohganz, Holger & Rades, Thomas, 4 Mar 2019, In: Molecular Pharmaceutics. 16, 3, p. 1294-1304 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    Whey proteins as stabilizers in amorphous solid dispersions

    Mishra, J., Bohr, A., Rades, Thomas, Grohganz, Holger & Löbmann, Korbinian, 1 Feb 2019, In: European Journal of Pharmaceutical Sciences. 128, p. 144-151 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Process Optimization and Upscaling of Spray-Dried Drug-Amino acid Co-Amorphous Formulations

    Kasten, G., Duarte, Í., Paisana, M., Löbmann, Korbinian, Rades, Thomas & Grohganz, Holger, 9 Jan 2019, In: Pharmaceutics. 11, 1, 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Characterising glass transition temperatures and glass dynamics in mesoporous silica-based amorphous drugs

    Kissi, E. O., Ruggiero, M. T., Hempel, N. J., Song, Z., Grohganz, Holger, Rades, Thomas & Löbmann, Korbinian, 1 Jan 2019, In: Physical Chemistry Chemical Physics. 21, 35, p. 19686-19694 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  51. Published

    Dipeptides as co-formers in co-amorphous systems

    Wu, W., Löbmann, Korbinian, Schnitzkewitz, J., Knuhtsen, A., Pedersen, D. S., Rades, Thomas & Grohganz, Holger, 1 Jan 2019, In: European Journal of Pharmaceutics and Biopharmaceutics. 134, p. 68-76 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  52. Published

    Influence of Glass Forming Ability on the Physical Stability of Supersaturated Amorphous Solid Dispersions

    Blaabjerg, L. I., Bulduk, B., Lindenberg, E., Löbmann, Korbinian, Rades, Thomas & Grohganz, Holger, 1 Jan 2019, In: Journal of Pharmaceutical Sciences. 108, 8, p. 2561-2569

    Research output: Contribution to journalJournal articleResearchpeer-review

  53. Published

    A co-amorphous form of a substance and a protein

    Mishra, J., Bohr, A., Berg, T. H. A., Löbmann, Korbinian, Rades, Thomas, Grohganz, Holger & Water, J. J., 2019, Patent No. US201903078886A1

    Research output: Patent

  54. Published

    Co-former selection for co-amorphous drug-amino acid formulations

    Kasten, G., Löbmann, Korbinian, Grohganz, Holger & Rades, Thomas, 2019, In: International Journal of Pharmaceutics. 557, p. 366-373

    Research output: Contribution to journalJournal articleResearchpeer-review

  55. Published

    Efflux Inhibitor Bicalutamide Increases Oral Bioavailability of the Poorly Soluble Efflux Substrate Docetaxel in Co-Amorphous Anti-Cancer Combination Therapy

    Bohr, A., Nascimento, T. L., Harmankaya, N., Weisser, J. J., Wang, Y., Grohganz, Holger, Rades, Thomas & Löbmann, Korbinian, 2019, In: Molecules. 24, 2, 13 p., 266.

    Research output: Contribution to journalJournal articleResearchpeer-review

  56. Published

    Impact of drug loading in mesoporous silica-amorphous formulations on the physical stability of drugs with high recrystallization tendency

    Antonino, R. S. C. M. Q., Ruggiero, M., Song, Z., Nascimento, T. L., Lima, E. M., Bohr, A., Knopp, Matthias Manne & Löbmann, Korbinian, 2019, In: International Journal of Pharmaceutics: X. 1, 7 p., 100026.

    Research output: Contribution to journalJournal articleResearchpeer-review

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