Birger Brodin Larsen
Professor
CNS Drug Delivery and Barrier Modelling
Universitetsparken 2
2100 København Ø
- 2008
- Published
Sorption and mobility of ivermectin in different soils
Krogh, K. A., Søborg, T., Larsen, Birger Brodin & Halling-Sørensen, B., 2008, In: Journal of Environmental Quality. 37, 6, p. 2202-2211Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Transport of amino acids and GABA analogues via the human proton-coupled amino acid transporter, hPAT1: Characterization of conditions for affinity and transport experiments in Caco-2 cells.
Larsen, M., Larsen, Birger Brodin, Frølund, Bente & Nielsen, C. U., 2008, In: European Journal of Pharmaceutical Sciences. 35, 1-2, p. 86-95Research output: Contribution to journal › Journal article › Research › peer-review
- Published
hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3
Søndergaard, H. B., Larsen, Birger Brodin & Nielsen, C. U., 2008, In: Pflügers Archiv: European Journal of Physiology. 456, 3, p. 611-622Research output: Contribution to journal › Journal article › Research › peer-review
- 2007
- Published
Basolateral peptide transport in intestinal cells is pH dependent
Juul Nielsen, M., Nielsen, C. U. & Larsen, Birger Brodin, 2007. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Molekylær biofarmaci - når medicinen skyder genvej!
Gram, L. K., Omkvist, D. H., Larsen, M., Nielsen, C. U., Larsen, Birger Brodin & Steffansen, I. D., 2007, In: Lægemiddelforskning. p. 16-17Research output: Contribution to journal › Journal article › Communication
- Published
Optimization of a cell-based flourescent probe assay for measuring substrate translocation via the proton-coupled intestinal di/tri-peptide transporter hPEPT1
Omkvist, D. H., Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, 2007. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Peptide Transporters in Drug Delivery
Larsen, Birger Brodin, Steffansen, B. & Nielsen, C. U., 2007. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Proton-coupled basolateral dipeptide transport in a human intestinal cell line, Caco-2
Larsen, Birger Brodin, Nielsen, M. J. & Nielsen, C. U., 2007. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
The human proton-coupled amino acid transporter (hPAT1) is a transport system for GABA-like drugs
Broberg, M. L., Frølund, Bente, Larsen, Birger Brodin & Nielsen, C. U., 2007. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- 2006
- Published
Genetic variants of the human dipeptide transporter PEPT1
Anderle, P., Nielsen, C. U., Pinsonneault, J., Krog, P. L., Larsen, Birger Brodin & Sadée, W., 1 Feb 2006, In: Journal of Pharmacology and Experimental Therapeutics. 316, 2, p. 636-646 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Carbonic anhydrase imhibitors. Transepithelial transport of novel anticancer sulfonamide inhibitors of the cancer-associated isozyme CA IX is dependent on the p.gp efflux transporter
Vullo, D., Steffansen, B., Larsen, Birger Brodin, Supuran, C. T., Scozzafava, A. & Nielsen, C. U., 2006, In: Bioorganic & Medicinal Chemistry Letters. 14, 7, p. 2418-2427Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Carrier-mediated dipeptide transport in a human lung epithelial cell line, Calu-3
Nielsen, C. U., Søndergaard, H. B. & Larsen, Birger Brodin, 2006. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1
Andersen, R., Nielsen, C. U., Begtrup, M., Jørgensen, Flemming Steen, Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2006, In: European Journal of Pharmaceutical Sciences. 28, 4, p. 325-35 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Insulin increases peptide transport capacity in the proximal tubule kidney cell line SKPT0193-Cl.2.
Rquez, B., Nielsen, C. U. & Larsen, Birger Brodin, 2006. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Oral Gly-Sar absorption is inhibited bu a high-affinity PEPT1 inhibitor Lys-Z-NO2-Pro
Eriksson, A. H., Rist, G. M., Larsen, Birger Brodin & Steffansen, B., 2006. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
Proton dependent transport of amino acids in Caco-2 cells
Broberg, M. L., Larsen, Birger Brodin & Nielsen, C. U., 2006. 1 p.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- 2005
- Published
Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media
Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 2, p. 98-108 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Particle size and surface charge affect particle uptake by human dendritic cells in an in vitro model
Foged, Camilla, Larsen, Birger Brodin, Frøkjær, Sven & Sundblad, A., 2005, In: Internation Journal of Pharmaceutics. 298, 2, p. 315-22 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Pyrimidine and nucleoside gamma-esters of L-Glu-Sar: synthesis, stability and interaction with hPEPT1
Eriksson, A. H., Elm, P. L., Begtrup, M., Larsen, Birger Brodin, Nielsen, R. & Steffansen, B., 2005, In: European Journal of Pharmaceutical Sciences. 25, 1, p. 145-154 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Recent advances in therapeutic applications of human transporters
Nielsen, C. U., Våbenø, J., Andersen, R., Larsen, Birger Brodin & Steffansen, B., 2005, In: Expert Opinion on Therapeutic Patents. 15, 2, p. 153-166 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The F28Y substitution in the human intestinal di/tri-peptide transporter hPEPT1, causes altered pH-dependency of Gly-Sar transport
Nielsen, C. U., Krog, P., Anderlee, P., Sadeé, W. & Larsen, Birger Brodin, 2005.Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
- Published
hPEPT1 Affinity and Translocation of Selected Gln-Sar and Glu-Sar Dipeptide Derivatives
Eriksson, A. H., Elm, P. L., Begtrup, M., Nielsen, R., Steffansen, B. & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 3, p. 242-249Research output: Contribution to journal › Journal article › Research › peer-review
- 2004
- Published
In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model
Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 1 Jan 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 77-86 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2
Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 2004, In: American Journal of Physiology - Renal Physiology. 286, 2, p. 385-393Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Intestinal solute carriers: an overview of trends and strategies for improving oral drug absorption
Steffansen, B., Nielsen, C. U., Larsen, Birger Brodin, Eriksson, A. H., Andersen, R. & Frøkjær, Sven, 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 3-16 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1299175
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Design of prodrugs targeting the intestinal di/tri‐peptide transporter hPEPT1 (SLC15A1
Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
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A bovine in vitro blood-brain barrier model under oxygenglucose deprivation (OGD) condition
Research output: Contribution to conference › Poster › Research
Published