Birger Brodin Larsen

Birger Brodin Larsen

Professor


  1. 2012
  2. Published

    In-vitro evaluation of the P-glycoprotein interactions of a series of potentially CNS-active Amaryllidaceae alkaloids

    Eriksson, A. H., Rønsted, Nina, Jäger, A. K., Sendra, J. R. & Larsen, Birger Brodin, 2012, In: Journal of Pharmacy and Pharmacology. 64, 11, p. 1667-1677 11 p.

    Research output: Contribution to journalJournal articlepeer-review

  3. Published

    In-vitro models of the blood brain barrier

    Larsen, Birger Brodin, Helms, H. C. C., Groth, S., Waagepetersen, Helle S. & Nielsen, C. U., 2012. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  4. Published

    Kostens sammensætning kan påvirke optagelsen af lægemiddelstoffer

    Nielsen, C. U., Frølund, S. B., Nøhr, M. K., Larsen, Birger Brodin & Holm, R., 2012, In: Lægemiddelforskning. 2012, p. 31-33

    Research output: Contribution to journalJournal article

  5. 2011
  6. Published

    Bovine endothelial/rat astrocyte co-cultures cultured in highly buffered media functionally express MDR1 and BCRP

    Helms, H. C. C., Badolo, L., Kuhlmann, L. B. & Larsen, Birger Brodin, 21 Jun 2011.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  7. Published

    Affinity and translocation relationships via hPEPT1 of H-Xaa-Ser-OH dipeptides: evaluation of H-Phe-Ser-OH as a pro-moiety for ibuprofen and benzoic acid prodrugs

    Omkvist, D. H., Trangbæk, D. J., Mildon, J., Paine, J. S., Larsen, Birger Brodin, Begtrup, M. & Nielsen, C. U., 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 77, 2, p. 327-331

    Research output: Contribution to journalJournal articlepeer-review

  8. Published

    Calu-3 cells grown under AIC and LCC conditions: implications for dipeptide uptake and transepithelial transport of substances

    Stentebjerg-Andersen, A., Notlevesen, I. V., Larsen, Birger Brodin & Nielsen, C. U., 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 78, 1, p. 19-26

    Research output: Contribution to journalJournal articlepeer-review

  9. Published

    Transport af lægemiddelstoffer gennem vævsbarrier

    Nielsen, C. U. & Larsen, Birger Brodin, 2011, Bioteknologi - en temabog. Gasbjerg, P. K., Jensen, G. S. & Sørensen, A. B. (eds.). Århus: Systime, p. 145-157 12 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterEducationpeer-review

  10. 2010
  11. Published

    Paracellular tightness and claudin-5 expression is increased in the BCEC/Astrocyte blood-brain barrier model by increasing media buffer capacity during growth

    Helms, H. C., Waagepetersen, Helle S., Nielsen, C. U. & Larsen, Birger Brodin, Dec 2010, In: The AAPS Journal. 12, 4, p. 759-770

    Research output: Contribution to journalJournal articlepeer-review

  12. Published

    Planternes slægtskab som skattekort til nye lægemidler

    Rønsted, Nina, Larsen, Birger Brodin, Christensen, Søren Brøgger, Eriksson, A. H. & Jäger, A. K., Dec 2010, In: Lægemiddelforskning. 2010, p. 19-21

    Research output: Contribution to journalJournal article

  13. Published

    The interaction of CNS-active Amaryllidae alkaloids with the BBB efflux pump MDR1

    Eriksson, A. H., Birrer, A., Sendra, J. R., Güler, S., Rønsted, Nina, Jäger, A. K. & Larsen, Birger Brodin, 29 Jun 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  14. Published

    Gly-Sar is a substrate for the human proton-coupled amino acid transporter, hPAT1 (SLC36A1)

    Frølund, S. B., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., Mar 2010.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  15. Published

    Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., Mar 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  16. Published

    mRNA expression and transport function of the proton-coupled amino acid transporter , PAT1, along the rat intestine

    Broberg, M. L., Brandt Larsen, K., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., Mar 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  17. Published

    5-Hydroxy-L-tryptohan alters gaboxadol pharmacokinetics in rats: involvement of PAT1 and rOat1 in gaboxadol absorption and elimination

    Broberg, M. L., Holm, R., Jensen, K. G., Sveigaard, C., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: European Journal of Pharmaceutical Sciences. 39, 1-3, p. 68-75

    Research output: Contribution to journalJournal articlepeer-review

  18. Published

    A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1)

    Omkvist, D. H., Larsen, S. B., Nielsen, C. U., Steffansen, B., Olsen, L., Jørgensen, Flemming Steen & Larsen, Birger Brodin, 2010, In: The AAPS Journal. 12, 3, p. 385-396

    Research output: Contribution to journalJournal articlepeer-review

  19. Published

    Absorptive transporters

    Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage from evaluation. Steffansen, B., Brodin, B. & Uhd Nielsen, C. (eds.). London: Pharmaceutical Press, p. 193-211 (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  20. Published

    Acid/base properties, solubility and distribution of drug candidates

    Steffansen, B., Nielsen, C. U. & Larsen, Birger Brodin, 2010, Molecular Biopharmaceutics: Aspects of drug characterization drug delivery and dosage form evaluation. Pharmaceutical Press, p. 5-31

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  21. Published

    Carrier-mediated transport kinetics

    Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Pharmaceutical Press, p. 153-173

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  22. Published

    Claudin-5 mRNA expression and transendothelial electrical resistance (TEER) correlate in the BCEC/astrocyte blood-brain barrier model

    Helms, H. C. C., Waagepetersen, Helle S., Nielsen, C. U. & Larsen, Birger Brodin, 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  23. Published

    Efflux transporters

    Nielsen, C. U., Larsen, Birger Brodin & Steffansen, B., 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Steffansen, B., Brodin, B. & Uhd Nielsen, C. (eds.). Pharmaceutical Press, p. 213-22

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  24. Published

    GABA transport across the basolateral membrane of intestinal cells

    Nielsen, C. U., Carstensen, M. & Larsen, Birger Brodin, 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  25. Published

    Gly-sar is a substrate for the human proton coupled amino acid trasporter 1, hPAT1 (SLC36A1)

    Frølund, S. B., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., 2010.

    Research output: Contribution to conferencePosterResearch

  26. Published

    Hjernens forsvarsmur kortlagt og kopieret

    Helms, H. C., Waagepetersen, Helle S., Nielsen, C. U. & Larsen, Birger Brodin, 2010, In: Lægemiddelforskning. 2010, p. 22-24

    Research output: Contribution to journalJournal article

  27. Published

    Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 161, 8, p. 1793-1805

    Research output: Contribution to journalJournal articlepeer-review

  28. Published

    Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010.

    Research output: Contribution to conferencePosterResearch

  29. Published

    In vitro models for investigating the function of proton-coupled amino acid transporter 1 (PAT1, SLC36A19)

    Jensen, A., Larsen, Birger Brodin & Nielsen, C. U., 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  30. Published

    Introduction

    Steffansen, B., Nielsen, C. U. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage from evaluation. Steffansen, B., Brodin, B. & Uhd Nielsen, C. (eds.). London: Pharmaceutical Press, p. 1-4 4 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  31. Published

    Kinetics of decomposition in aqueous solution

    Steffansen, B., Nielsen, C. U. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Steffansen, B., Brodin, B. & Nielsen, C. U. (eds.). Pharmaceutical Press, p. 51-69 (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  32. Published

    Mechanism of decomposition of drug candidates

    Steffansen, B., Nielsen, C. U. & Larsen, Birger Brodin, 2010, Molecular Biopharmaceutics: Aspects of drug characterization, drug delivery and dosage form evaluation. Pharmaceutical Press, p. 35-48 13 p. (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  33. Published

    Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation

    Steffansen, B., Larsen, Birger Brodin & Nielsen, C. U., 2010, Pharmaceutical Press. (ULLA Pharmacy Series).

    Research output: Book/ReportBookpeer-review

  34. Published

    Passive diffusion of drug substances: the concepts of flux and permeability

    Larsen, Birger Brodin, Steffansen, B. & Nielsen, C. U., 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Steffansen, B., Brodin, B. & Nielsen, C. U. (eds.). PharmaPress Ltd., p. 135-151 16 p. (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  35. Published

    Structure and function of absorption barriers

    Larsen, Birger Brodin, Steffansen, B. & Nielsen, C. U., 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Steffansen, B., Brodin, B. & Nielsen, C. U. (eds.). Pharmaceutical Press, p. 115-131 (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  36. Published

    The expression of Claudin-5 correlates with transendothelial electrical resistance (TEER) in BCEC/rat astrocyte blood-brain barrier models

    Helms, H. C. C., Waagepetersen, Helle S., Nielsen, C. U. & Larsen, Birger Brodin, 2010.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  37. Published

    The proton-coupled amino acid transporter, SLC36A1 (hPAT1), transports Gly-Gly, Gly-Sar and other Gly-Gly mimetics

    Frølund, S., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 161, 3, p. 589-600

    Research output: Contribution to journalJournal articlepeer-review

  38. Published

    d-Aminolevulinic acid is a substrate for the amino acid transporter SLC36A1 (hPAT1)

    Frølund, S., Marquez, O. C., Larsen, M., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 159, 6, p. 1339-1353

    Research output: Contribution to journalJournal articlepeer-review

  39. Published

    mRNA expression and transport function of the proton-coupled amino acid transporter, PAT1, along the rat intestine

    Broberg, M. L., Larsen, K. B., Holm, R., Larsen, Birger Brodin & Nielsen, C. U., 2010.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  40. 2009
  41. Published

    Characterization of in vitro blood-brain barrier models

    Helms, H. C. C., Eriksson, A. H., Nielsen, C. U., Waagepetersen, Helle S., Walls, Anne Byriel & Larsen, Birger Brodin, 9 Aug 2009. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  42. Published

    Characterization of in-vitro blood-brain barrier models

    Helms, H. C. C., Eriksson, A. H., Nielsen, C. U., Waagepetersen, Helle S. & Larsen, Birger Brodin, Aug 2009.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  43. Published

    Transport of Gaboxadol via hPAT1 and rOAT1 in the absence and presence of 5-HTP

    Broberg, M. L., Holm, R., Larsen, Birger Brodin, Jensen, K. G. & Nielsen, C. U., 29 Jul 2009. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  44. Published

    In vitro blood-brain barrier models

    Helms, H. C. C., Eriksson, A. H., Nielsen, C. U., Waagepetersen, Helle S. & Larsen, Birger Brodin, 18 Jul 2009.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  45. Published

    Peptide transporters in drug delivery; The human peptide transporter 1 (hPEPT1) translocates differently charged peptides in an electrogenic manner, indicating a varying proton coupling ration

    Omkvist, D. H., Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, May 2009. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  46. Published

    In Vitro cutaneous application of ISCOMs on human skin enhances delivery of hydrophobic model compounds through the stratum corneum

    Madsen, H. B., Ifversen, P., Madsen, F., Larsen, Birger Brodin, Hausser, I. & Nielsen, Hanne Mørck, 2009, In: The AAPS Journal. 11, 4, p. 728-739

    Research output: Contribution to journalJournal articlepeer-review

  47. Published

    Characterisation of in-vitro blood-brain barrier models

    Helms, H. C., Eriksson, A. H., Waagepetersen, Helle S. & Larsen, Birger Brodin, 2009.

    Research output: Contribution to conferencePosterResearch

  48. Published

    Discovery of ligands for the human intestinal di-/tripeptide transporter (hPEPT1) using af QSAR-assisted virtual screening strategy

    Larsen, S. B., Omkvist, D. H., Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B., Olsen, L. & Jørgensen, Flemming Steen, 2009, In: ChemMedChem. 4, 9, p. 1439-1445

    Research output: Contribution to journalJournal articlepeer-review

  49. Published

    Gaboxadol bliver absorberet via en aminosyretransportør

    Broberg, M. L., Holm, R., Jensen, K. G., Larsen, Birger Brodin & Nielsen, C. U., 2009, In: Lægemiddelforskning. p. 22-24

    Research output: Contribution to journalJournal article

  50. Published

    Intestinal gaboxadol absorption via PAT1 (SLC36A1): modified absorption in vivo following co-administration of L-tryptophan

    Larsen, M., Larsen, R., Jensen, K. G., Larsen, Birger Brodin & Nielsen, C. U., 2009, In: British Journal of Pharmacology. 157, p. 1380-1389

    Research output: Contribution to journalJournal articlepeer-review

  51. 2008
  52. Published

    Basolateral peptid etransport in the human intestinal cell line Caco-2 is proton-coupled

    Nielsen, M. J., Nielsen, C. U. & Larsen, Birger Brodin, 2008. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  53. Published

    Cloning of the pig PEPT2 (pPEPT2) and characterization of the effects of epidermal growth factor (EGF) on pPEPT2-mediated peptide uptake in the renal porcine cell line LLC-PK1

    Søndergaard, H. B., Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2008, In: European Journal of Pharmaceutical Sciences. 33, 4-5, p. 332-342

    Research output: Contribution to journalJournal articlepeer-review

  54. Published

    Comparison of drug transporter gene expression and functionality in Caco-2 cells from 10 different laboratories

    Hayeshi, R., Hilgendorf, C., Arthursson, P., Augustijns, P., Larsen, Birger Brodin, Dehertogh, P., Fisher, K., Fossati, L., Hovenkamp, E., Korjamo, T., Masungi, C., Maubon, N., Mols, R., Mullertz, Anette , Mönkkönen, J., O´Driscoll, C., Oppers-Tiemissen, H. M., Ragnarsson, E. G. E., Rooseboom, M. & Ungell, A., 2008, In: European Journal of Pharmaceutical Sciences. 35, 5, p. 383-396

    Research output: Contribution to journalJournal articlepeer-review

  55. Published

    Sorption and mobility of ivermectin in different soils

    Krogh, K. A., Søborg, T., Larsen, Birger Brodin & Halling-Sørensen, B., 2008, In: Journal of Environmental Quality. 37, 6, p. 2202-2211

    Research output: Contribution to journalJournal articlepeer-review

ID: 1299175