Birger Brodin Larsen

Birger Brodin Larsen

Professor


  1. 2006
  2. Published

    In vitro evaluation of N-methyl amide tripeptidomimetics as substrates for the human intestinal di-/tri-peptide transporter hPEPT1

    Andersen, R., Nielsen, C. U., Begtrup, M., Jørgensen, Flemming Steen, Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2006, In: European Journal of Pharmaceutical Sciences. 28, 4, p. 325-35 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Insulin increases peptide transport capacity in the proximal tubule kidney cell line SKPT0193-Cl.2.

    Rquez, B., Nielsen, C. U. & Larsen, Birger Brodin, 2006. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  4. Published

    Oral Gly-Sar absorption is inhibited bu a high-affinity PEPT1 inhibitor Lys-Z-NO2-Pro

    Eriksson, A. H., Rist, G. M., Larsen, Birger Brodin & Steffansen, B., 2006. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  5. Published

    Proton dependent transport of amino acids in Caco-2 cells

    Broberg, M. L., Larsen, Birger Brodin & Nielsen, C. U., 2006. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  6. 2005
  7. Published

    Characterization of rPEPT2-mediated Gly-Sar transport parameters in the rat kidney proximal tubule cell line SKPT-0193 cl.2 cultured in basic growth media

    Bravo, S. A., Nielsen, C. U., Frøkjær, Sven & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 2, p. 98-108 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Particle size and surface charge affect particle uptake by human dendritic cells in an in vitro model

    Foged, Camilla, Larsen, Birger Brodin, Frøkjær, Sven & Sundblad, A., 2005, In: Internation Journal of Pharmaceutics. 298, 2, p. 315-22 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Pyrimidine and nucleoside gamma-esters of L-Glu-Sar: synthesis, stability and interaction with hPEPT1

    Eriksson, A. H., Elm, P. L., Begtrup, M., Larsen, Birger Brodin, Nielsen, R. & Steffansen, B., 2005, In: European Journal of Pharmaceutical Sciences. 25, 1, p. 145-154 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Recent advances in therapeutic applications of human transporters

    Nielsen, C. U., Våbenø, J., Andersen, R., Larsen, Birger Brodin & Steffansen, B., 2005, In: Expert Opinion on Therapeutic Patents. 15, 2, p. 153-166 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    The F28Y substitution in the human intestinal di/tri-peptide transporter hPEPT1, causes altered pH-dependency of Gly-Sar transport

    Nielsen, C. U., Krog, P., Anderlee, P., Sadeé, W. & Larsen, Birger Brodin, 2005.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  12. Published

    hPEPT1 Affinity and Translocation of Selected Gln-Sar and Glu-Sar Dipeptide Derivatives

    Eriksson, A. H., Elm, P. L., Begtrup, M., Nielsen, R., Steffansen, B. & Larsen, Birger Brodin, 2005, In: Molecular Pharmaceutics. 2, 3, p. 242-249

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. 2004
  14. Published

    In-depth evaluation of Gly-Sar transport parameters as a function of culture time in the Caco-2 cell model

    Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 1 Jan 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 77-86 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Epidermal growth factor decreases PEPT2 transport capacity and expression in the rat kidney proximal tubule cell line SKPT0193 cl.2

    Bravo, S. A., Nielsen, C. U., Amstrup, J., Frøkjær, Sven & Larsen, Birger Brodin, 2004, In: American Journal of Physiology - Renal Physiology. 286, 2, p. 385-393

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Intestinal solute carriers: an overview of trends and strategies for improving oral drug absorption

    Steffansen, B., Nielsen, C. U., Larsen, Birger Brodin, Eriksson, A. H., Andersen, R. & Frøkjær, Sven, 2004, In: European Journal of Pharmaceutical Sciences. 21, 1, p. 3-16 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. 2003
  18. Published

    Erratum: Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: Affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism (Journal of Controlled Release (2003) 86 (279-292) PII: S0168365902004133)

    Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 7 Mar 2003, In: Journal of Controlled Release. 88, 2

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Di/tri-peptide transporters as drug delivery targets: regulation of transport under physiological and patho-physiological conditions

    Nielsen, C. U. & Larsen, Birger Brodin, 2003, In: Current Drug Targets. 4, 5, p. 373-88 16 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Epidermal growth factor and insulin short-term increase hPEPT1-mediated glycylsarcosine uptake in Caco-2 cells

    Larsen, Birger Brodin, Amstrup, J., Nielsen, C. U., Steffansen, B. & Frøkjær, S., 2003, In: Acta Physiol. Scandinavia. 178, p. 139-148

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism

    Thomsen, A. E., Friedrichsen, G. M., Sørensen, A. H., Andersen, R., Nielsen, C. U., Larsen, Birger Brodin, Begtrup, M., Frøkjær, Sven & Steffansen, B., 2003, In: Journal of Controlled Release. 86, 2-3, p. 279-92 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. 2002
  23. Published

    Human peptide transporters: Therapeutic applications

    Nielsen, C. U., Larsen, Birger Brodin, Jørgensen, Flemming Steen, Frøkjær, Sven & Steffansen, B., 1 Sep 2002, In: Expert Opinion on Therapeutic Patents. 12, 9, p. 1329-1350 22 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Transport characteristics of L-carnosine and the anticancer derivative 4-toluenesulfonylureido-carnosine in a human epithelial cell line

    Nielsen, C. U., Supuran, C. T., Scozzafava, A., Frøkjær, Sven, Steffansen, B. & Larsen, Birger Brodin, 2002, In: Pharmaceutical Research. 19, 9, p. 1337-44 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Transport of peptidomimetic drugs by the intestinal Di/tri-peptide transporter, PepT1

    Larsen, Birger Brodin, Nielsen, C. U., Steffansen, B. & Frøkjær, Sven, 2002, In: Basic & Clinical Pharmacology & Toxicology. 90, 6, p. 285-96 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. 2001
  27. Published

    Cloning and characterization of a human orphan family C G-protein coupled receptor GPRC5D

    Bräuner, Hans, Jensen, Anders A., Sheppard, P. O., Larsen, Birger Brodin, Krogsgaard-Larsen, Povl & O'Hara, P., 2001, In: BBA General Subjects. 1518, 3, p. 237-48 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line

    Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven, Taub, M. E. & Steffansen, B., 2001, In: Journal of Controlled Release. 76, 1-2, p. 129-38 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Epidermal growth factor inhibits glycylsarcosine transport and hPepT1 expression in a human intestinal cell line

    Nielsen, C. U., Amstrup, J., Steffansen, B., Frøkjær, Sven & Larsen, Birger Brodin, 2001, In: American Journal of Physiology: Gastrointestinal and Liver Physiology. 281, 1, p. G191-9

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Model prodrugs for the intestinal oligopeptide transporter: model drug release in aqueous solution and in various biological media

    Nielsen, C. U., Andersen, R., Larsen, Birger Brodin, Frøkjær, Sven & Steffansen, B., 2001, In: Journal of Controlled Release. 73, 1, p. 21-30 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. 2000
  32. Published

    Evidence for P2Y-type ATP receptors on the serosal membrane of frog skin epithelium

    Larsen, Birger Brodin & Nielsen, R., 1 Jan 2000, In: Pflugers Archiv European Journal of Physiology. 439, 3, p. 234-239 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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